SCHEMBL7042013

SCHEMBL7042013

NC(=O)c1cccc2ncc(-c3ccc([N+](=O)[O-])cc3)nc12

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.71
PARP2 Q9UGN5 1/20 0.67
NPC1 O15118 5/20 0.60
RAB9A P51151 4/20 0.60
CASP1 P29466 1/20 0.48
MAPT P10636 4/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
LMNA P02545 2/20 0.43
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7040069 0.88 NPC1 (0.64) PARP1PARP2NPC1RAB9AMAPT
SCHEMBL7112515 0.83 PARP1 (1.00) PARP1PARP2NPC1RAB9A
SCHEMBL7111338 0.83 PARP1 (0.80) PARP1PARP2ALDH1A1
SCHEMBL424209 0.82 PARP1 (0.81) PARP1PARP2NPC1RAB9ACASP1
SCHEMBL7045309 0.82 PARP1 (0.78) PARP1PARP2ALDH1A1
SCHEMBL31602072 0.82 PARP1 (0.81) PARP1PARP2NPC1RAB9ACASP1
SCHEMBL7042977 0.82 PARP1 (0.78) PARP1PARP2CASP1KMT2A
SCHEMBL7108289 0.80 PARP1 (1.00) PARP1PARP2CASP1
SCHEMBL7107333 0.79 PARP1 (1.00) PARP1PARP2CASP1
SCHEMBL7045177 0.79 PARP1 (1.00) PARP1PARP2NPC1RAB9ACASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed