SCHEMBL7040069

SCHEMBL7040069

NC(=O)c1cccc2ncc(-c3cccc([N+](=O)[O-])c3)nc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.64
RAB9A P51151 4/20 0.64
PARP1 P09874 6/20 0.61
BCHE P06276 1/20 0.59
ACHE P22303 1/20 0.59
PARP2 Q9UGN5 1/20 0.58
MAPT P10636 4/20 0.52
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 1/20 0.47
CYP1A2 P05177 1/20 0.47
TOP1 P11387 1/20 0.47
CDC7 O00311 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
KCNH2 Q12809 1/20 0.46
THRB P10828 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
IDO1 P14902 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4C Q08493 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042013 0.88 PARP1 (0.71) NPC1RAB9APARP1BCHEACHE
SCHEMBL7111338 0.81 PARP1 (0.80) PARP1PARP2ALDH1A1
SCHEMBL7113559 0.81 PARP1 (0.67) NPC1RAB9APARP1BCHEACHE
SCHEMBL7043497 0.79 PARP1 (0.71) PARP1PARP2KMT2A
SCHEMBL1463396 0.79 NPC1 (1.00) NPC1RAB9ABCHEACHEMAPT
SCHEMBL7046986 0.78 PARP1 (0.70) PARP1PARP2CDC7
SCHEMBL7115056 0.78 PARP1 (0.78) PARP1PARP2MAPTCYP1A2TOP1
SCHEMBL7045348 0.77 PARP1 (0.69) PARP1PARP2MAPT
SCHEMBL7112515 0.76 PARP1 (1.00) NPC1RAB9APARP1PARP2
SCHEMBL28222646 0.76 RAB9A (0.70) NPC1RAB9ABCHEACHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed