SCHEMBL7043497

SCHEMBL7043497

NC(=O)c1cccc2ncc(-c3cccnc3)nc12

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.71
PARP2 Q9UGN5 2/20 0.67
PKN1 Q16512 1/20 0.57
PKN2 Q16513 1/20 0.57
DHODH Q02127 1/20 0.54
KMT2A Q03164 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
MKNK1 Q9BUB5 5/20 0.48
MKNK2 Q9HBH9 4/20 0.48
MAPK1 P28482 2/20 0.47
ATR Q13535 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7111338 0.89 PARP1 (0.80) PARP1PARP2PKN1PKN2DHODH
SCHEMBL7112515 0.83 PARP1 (1.00) PARP1PARP2PKN1PKN2DHODH
SCHEMBL20660475 0.83 PARP1 (0.60) PARP1PARP2KMT2AATR
SCHEMBL7113559 0.83 PARP1 (0.67) PARP1PARP2KMT2ARXFP1
SCHEMBL7042977 0.82 PARP1 (0.78) PARP1PARP2DHODHKMT2ARXFP1
SCHEMBL424209 0.82 PARP1 (0.81) PARP1PARP2DHODHKMT2AATR
SCHEMBL31602072 0.82 PARP1 (0.81) PARP1PARP2DHODHKMT2AATR
SCHEMBL7045309 0.82 PARP1 (0.78) PARP1PARP2DHODHMAPK1ATR
SCHEMBL7108289 0.80 PARP1 (1.00) PARP1PARP2ATR
SCHEMBL7046986 0.80 PARP1 (0.70) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO claimed
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed