SCHEMBL7048978

SCHEMBL7048978

O=C(NCc1ccccc1F)Nc1nc2cc(OS(=O)(=O)c3ccc(-n4ccnc4)cc3)ccc2[nH]1.O=C(NCc1ccccc1F)Nc1nc2cc(OS(=O)(=O)c3ccc(NC4CCCC4)cc3)ccc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACR P10323 1/20 0.41
NAMPT P43490 3/20 0.39
MET P08581 1/20 0.39
CDK9 P50750 1/20 0.39
MCHR1 Q99705 4/20 0.36
NOS2 P35228 1/20 0.35
ROCK2 O75116 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
LMNA P02545 1/20 0.34
MMP1 P03956 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SLC6A9 P48067 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5042867 0.92 ACR (0.47) ACRNAMPTMETCDK9MCHR1
SCHEMBL5042907 0.92 ACR (0.48) ACRNAMPTMETCDK9NPC1
SCHEMBL7046318 0.87 RAB9A (0.39) NAMPTNOS2ROCK2NPC1RAB9A
SCHEMBL7045648 0.85 MEN1 (0.38) METCDK9NPC1RAB9ALMNA
SCHEMBL7176912 0.84 MAPT (0.39) METCDK9ROCK2NPC1RAB9A
SCHEMBL7044404 0.84 ROCK2 (0.37) NOS2ROCK2NPC1RAB9AMMP1
SCHEMBL7049236 0.84 MMP1 (0.38) NOS2ROCK2NPC1RAB9ALMNA
SCHEMBL5037966 0.84 MET (0.40) ACRNAMPTMETCDK9LMNA
SCHEMBL7044049 0.83 KDR (0.41) METCDK9ROCK2NPC1RAB9A
SCHEMBL5033564 0.83 MET (0.40) ACRNAMPTMETCDK9ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432417-A2 SUBSTITUTED BENZIMIDAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCER Aventis Pharma S.A. (FR) 2004-06-30 EP disclosed
WO-2003028721-A2 SUBSTITUTED BENZIMIDAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCER AVENTIS PHARMA S.A. (FR) 2003-04-10 WO disclosed