SCHEMBL7054866

SCHEMBL7054866

ClCO[CH]c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
MAOB P27338 2/20 0.36
TSHR P16473 1/20 0.36
CYP2A6 P11509 1/20 0.36
IDO1 P14902 2/20 0.35
ESR1 P03372 1/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
RELA Q04206 1/20 0.33
TRPA1 O75762 1/20 0.32
CYP19A1 P11511 2/20 0.31
CYP11B2 P19099 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PAM P19021 1/20 0.31
NFE2L2 Q16236 1/20 0.31
MAOA P21397 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9798232 0.79 ALDH1A1 (0.39) ALDH1A1MAOBTSHRCYP2A6IDO1
SCHEMBL3657712 0.78 KCNA3 (0.38) IDO1RELA
SCHEMBL10385527 0.76 MAOB (0.50) ALDH1A1MAOBIDO1LMNARELA
SCHEMBL93706 0.75 RELA (0.47) ALDH1A1MAOBTSHRCYP2A6IDO1
SCHEMBL2769032 0.75 ALDH1A1 (0.36) ALDH1A1MAOBTSHRCYP2A6IDO1
SCHEMBL9217606 0.75 ALDH1A1 (0.36) ALDH1A1MAOBTSHRCYP2A6IDO1
SCHEMBL790911 0.75 ALDH1A1 (0.36) ALDH1A1MAOBTSHRCYP2A6IDO1
SCHEMBL29135403 0.75 IDO1 (0.36) ALDH1A1MAOBTSHRCYP2A6IDO1
SCHEMBL8697137 0.74 KMT2A (0.32) ALDH1A1LMNAMEN1KMT2A
SCHEMBL425560 0.73 TSHR (0.50) ALDH1A1MAOBTSHRIDO1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1304325-A1 5-(M-CYANOBENZYLAMINO)PYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-04-23 EP disclosed
EP-0929535-A4 PROCESS AND NOVEL INTERMEDIATES LILLY CO ELI (US) 2001-05-23 EP disclosed
EP-0792875-B1 Cryptophycin derivatives and their use as anti-microtubule agents LILLY CO ELI (US) 2001-05-09 EP disclosed
EP-0929535-A1 PROCESS AND NOVEL INTERMEDIATES ELI LILLY AND COMPANY (US) 1999-07-21 EP disclosed
WO-1998009955-A1 PROCESS AND NOVEL INTERMEDIATES ELI LILLY AND COMPANY (US) 1998-03-12 WO disclosed
EP-0792875-A1 Cryptophycin derivatives and their use as anti-microtubule agents ELI LILLY AND COMPANY (US) 1997-09-03 EP disclosed
EP-0735819-A4 NEW CRYPTOPHYCINS UNIV HAWAII (US) 1997-03-19 EP disclosed
EP-0735819-A1 NEW CRYPTOPHYCINS UNIVERSITY OF HAWAII (US) 1996-10-09 EP disclosed
WO-1995017093-A1 NEW CRYPTOPHYCINS UNIVERSITY OF HAWAII (US) 1995-06-29 WO disclosed
US-4678792-A ANTITHROMBIC AGENTS DR. KARL THOMAE GMBH (DE) 1987-07-07 US disclosed
EP-0154842-A2 Medicament containing quaternary 3,4-dihydroisoquinoline salts Dr. Karl Thomae GmbH (DE) 1985-09-18 EP disclosed