SCHEMBL9217606

SCHEMBL9217606

BrCO[CH]c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
TSHR P16473 2/20 0.36
TRPA1 O75762 2/20 0.36
MAOB P27338 1/20 0.36
CYP2A6 P11509 1/20 0.36
IDO1 P14902 2/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TDP1 Q9NUW8 1/20 0.33
RELA Q04206 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
AKR1C3 P42330 1/20 0.32
PAM P19021 1/20 0.31
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9798232 0.79 ALDH1A1 (0.39) ALDH1A1TSHRTRPA1MAOBCYP2A6
SCHEMBL25245587 0.76 MAOB (0.44) ALDH1A1TRPA1MAOBIDO1LMNA
SCHEMBL790911 0.75 ALDH1A1 (0.36) ALDH1A1TSHRMAOBCYP2A6IDO1
SCHEMBL29135403 0.75 IDO1 (0.36) ALDH1A1TSHRTRPA1MAOBCYP2A6
SCHEMBL7054866 0.75 ALDH1A1 (0.36) ALDH1A1TSHRTRPA1MAOBCYP2A6
SCHEMBL2769032 0.75 ALDH1A1 (0.36) ALDH1A1TSHRTRPA1MAOBCYP2A6
SCHEMBL93706 0.75 RELA (0.47) ALDH1A1TSHRTRPA1MAOBCYP2A6
SCHEMBL425560 0.73 TSHR (0.50) ALDH1A1TSHRMAOBIDO1LMNA
SCHEMBL635906 0.71 TAAR1 (0.46) ALDH1A1TSHRCYP2A6IDO1TDP1
SCHEMBL5410674 0.71 TRPA1 (0.39) ALDH1A1TSHRTRPA1MAOBIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354788-B1 Novel imidazole derivatives NIPPON CHEMIPHAR CO (JP) 1995-09-13 EP disclosed
US-5180836-A Antiulcer agents NIPPON CHEMIPHAR CO., LTD. (JP) 1993-01-19 US disclosed
US-5082943-A Antiulcer NIPPON CHEMIPHAR CO., LTD. (JP) 1992-01-21 US disclosed
EP-0354788-A1 Novel imidazole derivatives NIPPON CHEMIPHAR CO., LTD. (JP) 1990-02-14 EP disclosed
US-4678792-A ANTITHROMBIC AGENTS DR. KARL THOMAE GMBH (DE) 1987-07-07 US disclosed
EP-0154842-A2 Medicament containing quaternary 3,4-dihydroisoquinoline salts Dr. Karl Thomae GmbH (DE) 1985-09-18 EP disclosed