SCHEMBL7065334

SCHEMBL7065334

CC(C)(C)OC[C@H]1O[C@](n2cnc3c(NC(=O)c4ccccc4)ncnc32)([SiH](c2ccccc2)c2ccccc2)[C@H](OCCO)[C@@H]1O

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 2/20 0.35
PRMT6 Q96LA8 1/20 0.34
ADORA1 P30542 6/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
P2RY2 P41231 1/20 0.33
P2RY1 P47900 1/20 0.33
P2RY6 Q15077 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7063493 0.93 P2RY12 (0.34) P2RY12PRMT6ADORA1ADORA3ADORA2A
SCHEMBL7251215 0.91 P2RY12 (0.34) P2RY12PRMT6ADORA1ADORA3ADORA2A
SCHEMBL7251726 0.91 P2RY12 (0.33) P2RY12PRMT6ADORA1ADORA3ADORA2A
SCHEMBL7063477 0.86 ADORA1 (0.46) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL7251671 0.83 P2RY12 (0.34) P2RY12PRMT6P2RY2P2RY1P2RY6
SCHEMBL7863923 0.80 PRMT6 (0.35) P2RY12PRMT6ADORA1ADORA3ADORA2A
SCHEMBL7064863 0.80 KDM4E (0.39)
SCHEMBL7063505 0.79 HINT1 (0.38) ADORA3
SCHEMBL6402247 0.78 ADORA1 (0.39) P2RY12ADORA1ADORA3ADORA2AADORA2B
SCHEMBL7246182 0.77 PRMT6 (0.33) PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6624294-B2 Dissolving nucleoside in solvent to form a solution; cooling; treating with base; warming; reacting with ester to effect alkylation of 2' position of a 2',3'-dihydroxy sugar moiety of a nucleoside ISIS PHARMACEUTICALS, INC. 2003-09-23 US disclosed
US-20030078415-A1 Regioselective synthesis of 2'-O-modified nucleosides IONIS PHARMACEUTICALS, INC. 2003-04-24 US disclosed
US-6403779-B1 DISSOLVING NUCLEOSIDE IN APROTIC SOLVENT, COOLING, TREATING WITH BASE, WARMING MIXTURE, COOLING, REACTING WITH REACTIVE ESTER TO EFFECT ALKYLATION ISIS PHARMACEUTICALS, INC. 2002-06-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078415-A1 Regioselective synthesis of 2'-O-modified nucleosides NSUN2, NT5C3B, RNGTT P2RY12 4230/4885PRMT6 1822/4885ADORA1 1499/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.