SCHEMBL7068296

SCHEMBL7068296

Cc1ccc(O/N=C\c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
PPARG P37231 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 2/20 0.41
LMNA P02545 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
PLA2G7 Q13093 1/20 0.41
VCAM1 P19320 1/20 0.40
EGFR P00533 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
GAA P10253 2/20 0.40
CYP1B1 Q16678 1/20 0.40
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12018747 0.86 LMNA (0.50) FAAHNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL2290696 0.86 LMNA (0.50) FAAHNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL2290693 0.86 LMNA (0.50) FAAHNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL29102043 0.74 ACHE (0.46) NPC1RAB9ASMN1; SMN2MAPTLMNA
SCHEMBL14336979 0.73 NPC1 (0.44) NPC1RAB9ASMN1; SMN2MAPTGAA
SCHEMBL14336940 0.73 RAB9A (0.44) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL14337015 0.72 VCAM1 (0.35) FAAHNPC1RAB9AMAPTLMNA
SCHEMBL14336980 0.72 VCAM1 (0.35) FAAHNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL3279914 0.70 ALDH1A1 (0.47) NPC1RAB9APPARGSMN1; SMN2MAPT
SCHEMBL113602 0.70 LMNA (0.52) FAAHNPC1RAB9APPARGSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066248-B1 METHYL-BIPHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI SYNTHELABO (FR) 2003-06-18 EP claimed
US-6417400-B1 O-(P-TOLYL)-BENZALDIMINE IS REACTED WITH HYDROXYLAMINE SALT TO FORM O-(P-TOLYL)-BENZALDOXIME; O-(P-TOLYL)-BENZONITRILE CHEMICAL INTERMEDIATES FOR DRUGS; OXIMINATION, IMINATION SANOFI-SYNTHELABO (FR) 2002-07-09 US claimed
EP-1066248-B1 METHYL-BIPHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI SYNTHELABO (FR) 2003-06-18 EP disclosed
EP-1066248-B1 METHYL-BIPHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI SYNTHELABO (FR) 2003-06-18 EP disclosed
US-6417400-B1 O-(P-TOLYL)-BENZALDIMINE IS REACTED WITH HYDROXYLAMINE SALT TO FORM O-(P-TOLYL)-BENZALDOXIME; O-(P-TOLYL)-BENZONITRILE CHEMICAL INTERMEDIATES FOR DRUGS; OXIMINATION, IMINATION SANOFI-SYNTHELABO (FR) 2002-07-09 US disclosed
US-6417400-B1 O-(P-TOLYL)-BENZALDIMINE IS REACTED WITH HYDROXYLAMINE SALT TO FORM O-(P-TOLYL)-BENZALDOXIME; O-(P-TOLYL)-BENZONITRILE CHEMICAL INTERMEDIATES FOR DRUGS; OXIMINATION, IMINATION SANOFI-SYNTHELABO (FR) 2002-07-09 US disclosed
EP-1066248-A1 METHYL-PHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI-SYNTHELABO (FR) 2001-01-10 EP disclosed
EP-1066248-A1 METHYL-PHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI-SYNTHELABO (FR) 2001-01-10 EP disclosed
WO-1999048861-A1 METHYL-PHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI-SYNTHELABO (FR) 1999-09-30 WO disclosed
WO-1999048861-A1 METHYL-PHENYL DERIVATIVES, PREPARATION METHOD AND USE SANOFI-SYNTHELABO (FR) 1999-09-30 WO disclosed