SCHEMBL7074575

SCHEMBL7074575

CCCCCCCCCCS(=O)(=O)N1CCN(C(=O)Cc2ccc(-c3noc(C)n3)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
DGAT1 O75907 1/20 0.47
JAK1 P23458 2/20 0.43
SPHK2 Q9NRA0 3/20 0.42
LMNA P02545 3/20 0.40
TSHR P16473 3/20 0.40
NPC1 O15118 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
PLA2G2A P14555 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR5 Q9H228 1/20 0.39
THRB P10828 1/20 0.39
SPHK1 Q9NYA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8080502 0.89 LMNA (0.44) DGAT1SPHK2LMNATSHRALDH1A1
SCHEMBL7077520 0.87 LMNA (0.54) HDAC4HDAC6LMNATSHRNPC1
SCHEMBL7074627 0.84 TSHR (0.57) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7074862 0.83 DGAT1 (0.53) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7074802 0.81 HDAC4 (0.53) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7071584 0.81 GAA (0.52) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7076669 0.81 GAA (0.53) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7069975 0.80 GAA (0.60) HDAC4HDAC6DGAT1LMNATSHR
SCHEMBL7075151 0.78 HDAC4 (0.49) HDAC4HDAC6DGAT1LMNANPC1
SCHEMBL7074530 0.78 THRB (0.52) DGAT1LMNANPC1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed