SCHEMBL7076517

SCHEMBL7076517

CN(Cc1cc2ccccc2o1)S(=O)(=O)Cc1ccccc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 6/20 0.43
MEN1 O00255 5/20 0.43
MAOB P27338 2/20 0.42
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
CA3 P07451 1/20 0.42
TSHR P16473 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
GPR35 Q9HC97 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
GALK1 P51570 1/20 0.42
NPC1 O15118 4/20 0.40
RAB9A P51151 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7072305 0.88 HDAC3 (0.42) ALDH1A1HPGDKMT2AMEN1MAOB
SCHEMBL7077693 0.88 RAB9A (0.49) ALDH1A1HPGDKMT2AMEN1NPC1
SCHEMBL7074387 0.75 ALDH1A1 (0.44) ALDH1A1HPGDKMT2AMEN1NPC1
SCHEMBL10683863 0.73 FOLH1 (0.47) ALDH1A1CA12CA9CA1TSHR
SCHEMBL7076158 0.70 MMP2 (0.44) ALDH1A1HPGDKMT2AMEN1NPC1
SCHEMBL15123483 0.68 CCR2 (0.62)
SCHEMBL7076161 0.67 ALDH1A1 (0.41) ALDH1A1HPGDKMT2AMEN1NPC1
SCHEMBL2393157 0.67 LOXL2 (0.53) ALDH1A1HPGDKMT2AMEN1MAOB
SCHEMBL3437042 0.66 KDM4E (0.48) ALDH1A1KMT2ACA9CA1TSHR
SCHEMBL1272937 0.66 LOXL2 (0.55) ALDH1A1HPGDMAOBCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003525203-A 2003-08-26 JP claimed
US-20030022893-A1 Hydroxamic and carboxylic acid derivatives BAXTER ANDREW DOUGLAS (GB) 2003-01-30 US claimed
EP-1163213-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES Darwin Discovery Limited (GB) 2001-12-19 EP claimed
WO-2000056704-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES DARWIN DISCOVERY LIMITED (GB) 2000-09-28 WO claimed
US-20030022893-A1 Hydroxamic and carboxylic acid derivatives BAXTER ANDREW DOUGLAS (GB) 2003-01-30 US disclosed
US-6465468-B1 SUCH AS N-HYDROXY-2-(4-(4-CHLOROPHENYL)PIPERAZINE-1-SULFONYL)BENZAMIDE; INHIBITORS OF MATRIX METALLOPROTEINASE, ADAM OR ADAMTS ENZYMES; TREATMENT OF DEGENERATIVE DISEASES AND CERTAIN CANCERS DARWIN DISCOVERY LIMITED (GB) 2002-10-15 US disclosed
EP-1163213-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES Darwin Discovery Limited (GB) 2001-12-19 EP disclosed
WO-2000056704-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES DARWIN DISCOVERY LIMITED (GB) 2000-09-28 WO disclosed