SCHEMBL7077693

SCHEMBL7077693

COC(=O)c1ccccc1CS(=O)(=O)N(C)Cc1cc2ccccc2o1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.49
NPC1 O15118 5/20 0.49
ALDH1A1 P00352 4/20 0.47
HPGD P15428 3/20 0.47
KDM4E B2RXH2 3/20 0.47
ATM Q13315 1/20 0.43
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
LMNA P02545 3/20 0.40
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
PPARG P37231 1/20 0.39
NCOA2 Q15596 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CASP3 P42574 1/20 0.38
SENP7 Q9BQF6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7076517 0.88 ALDH1A1 (0.44) RAB9ANPC1ALDH1A1HPGDKMT2A
SCHEMBL7072305 0.87 HDAC3 (0.42) RAB9ANPC1ALDH1A1HPGDKDM4E
SCHEMBL646787 0.75 L3MBTL1 (0.54) ALDH1A1KDM4EATMKMT2ALMNA
SCHEMBL15123480 0.73 CCR2 (0.60)
SCHEMBL7074387 0.70 ALDH1A1 (0.44) RAB9ANPC1ALDH1A1HPGDKMT2A
SCHEMBL7076158 0.70 MMP2 (0.44) RAB9ANPC1ALDH1A1HPGDKMT2A
SCHEMBL4880583 0.69 CA1 (0.58) ALDH1A1KDM4EATMKMT2ALMNA
SCHEMBL2383240 0.69 RAB9A (0.53) RAB9ANPC1ALDH1A1HPGDKDM4E
SCHEMBL8747734 0.69 KMT2A (0.57) ALDH1A1KDM4EKMT2AMEN1LMNA
SCHEMBL15123081 0.68 CCR2 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030022893-A1 Hydroxamic and carboxylic acid derivatives BAXTER ANDREW DOUGLAS (GB) 2003-01-30 US disclosed
US-6465468-B1 SUCH AS N-HYDROXY-2-(4-(4-CHLOROPHENYL)PIPERAZINE-1-SULFONYL)BENZAMIDE; INHIBITORS OF MATRIX METALLOPROTEINASE, ADAM OR ADAMTS ENZYMES; TREATMENT OF DEGENERATIVE DISEASES AND CERTAIN CANCERS DARWIN DISCOVERY LIMITED (GB) 2002-10-15 US disclosed