SCHEMBL7076841

SCHEMBL7076841

Cc1nc(-c2ccc(C(=O)N3CCN(OC(=O)Nc4ccccc4)CC3)cc2)no1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.54
DGAT1 O75907 3/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
HPGD P15428 1/20 0.47
HDAC4 P56524 3/20 0.46
GAA P10253 2/20 0.45
PLK1 P53350 1/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
MAPT P10636 4/20 0.44
MAPK14 Q16539 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074246 0.89 LMNA (0.52) MGLLLMNAHTTHPGDGAA
SCHEMBL7070524 0.88 STAT3 (0.52) LMNAHTTHPGDHDAC4HDAC2
SCHEMBL7073874 0.87 MAPT (0.52) MGLLLMNAHTTHPGDHDAC4
SCHEMBL7649408 0.86 DGAT1 (0.58) MGLLDGAT1LMNAHDAC4GAA
SCHEMBL7070301 0.86 MGLL (0.52) MGLLDGAT1LMNAHPGDHDAC4
SCHEMBL7071875 0.86 MAPT (0.51) MGLLLMNAHTTHPGDGAA
SCHEMBL7074772 0.83 MGLL (0.66) MGLLDGAT1LMNAHPGDHDAC4
SCHEMBL7077120 0.81 MGLL (0.47) MGLLDGAT1LMNAHDAC4PLK1
SCHEMBL7071622 0.80 SMYD3 (0.50) MGLLLMNAHDAC4PLK1HDAC2
SCHEMBL7074106 0.78 HDAC4 (0.58) MGLLDGAT1LMNAHTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed