SCHEMBL7076863

SCHEMBL7076863

CCCc1ccc(S(=O)(=O)N2CCN(Cc3ccc(-c4noc(C)n4)cc3)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 2/20 0.49
S1PR4 O95977 1/20 0.48
S1PR1 P21453 1/20 0.48
S1PR3 Q99500 1/20 0.48
S1PR5 Q9H228 1/20 0.48
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
ADORA2B P29275 2/20 0.46
ADORA3 P0DMS8 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 1/20 0.45
MAPK1 P28482 1/20 0.45
TSHR P16473 2/20 0.45
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7069980 0.89 TSHR (0.54) LSSCA12CA1CA2CA9
SCHEMBL7070226 0.88 THRB (0.54) CA12CA1CA2CA9ADORA2B
SCHEMBL7075159 0.87 LSS (0.51) LSSCA12CA1CA2CA9
SCHEMBL7074079 0.87 ALDH1A1 (0.63) ADORA2BTDP1SMN1; SMN2ALDH1A1LMNA
SCHEMBL7070564 0.85 LMNA (0.49) SMN1; SMN2ALDH1A1LMNAMAPK1MAPT
SCHEMBL7071584 0.84 GAA (0.52) CA12CA1CA2CA9SMN1; SMN2
SCHEMBL7074071 0.84 KDM4E (0.56) SMN1; SMN2ALDH1A1LMNATSHRMAPT
SCHEMBL8075470 0.84 LMNA (0.46) SMN1; SMN2ALDH1A1LMNAMAPT
SCHEMBL7076926 0.83 LSS (0.52) LSSTDP1SMN1; SMN2ALDH1A1LMNA
SCHEMBL7392302 0.82 LMNA (0.44) S1PR4S1PR1S1PR3S1PR5CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed