SCHEMBL7083490

SCHEMBL7083490

CNC(=S)OCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.35
GRIN2B Q13224 7/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
S1PR3 Q99500 4/20 0.33
ENPP2 Q13822 1/20 0.32
LMNA P02545 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
ATM Q13315 1/20 0.31
SRC P12931 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974277 0.94 GRIN1 (0.34) GRIN1GRIN2BS1PR3ENPP2TLR7
SCHEMBL6967842 0.91 ENPP2 (0.33) GRIN1GRIN2BENPP2LMNA
SCHEMBL7086281 0.90 ENPP2 (0.38) GRIN1GRIN2BS1PR3ENPP2LMNA
SCHEMBL7085898 0.90 ALDH1A1 (0.37) GRIN1GRIN2BGAAKMT2AS1PR3
SCHEMBL6976430 0.90 HTT (0.34) GAAS1PR3TLR7HTTSMN1; SMN2
SCHEMBL6972338 0.88 GRIN1 (0.38) GRIN1GRIN2BKMT2AS1PR3ENPP2
SCHEMBL6962639 0.88 RXFP1 (0.37) GAALMNAHTTSMN1; SMN2KDM4E
SCHEMBL7080182 0.87 MAPT (0.35) GRIN1GRIN2BKMT2AS1PR3HTT
SCHEMBL6969443 0.85 DHODH (0.32)
SCHEMBL6961326 0.85 GRIN1 (0.39) GRIN1GRIN2BGAAKMT2AS1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed