SCHEMBL7080360

SCHEMBL7080360

C=Cc1ccc(S(=O)(=O)NC2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
PKM P14618 2/20 0.52
HTT P42858 2/20 0.52
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
ALDH1A1 P00352 3/20 0.48
CCR6 P51684 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 1/20 0.47
HTR1A P08908 1/20 0.47
HTR7 P34969 1/20 0.47
TGM2 P21980 1/20 0.46
TP53 P04637 1/20 0.46
XBP1 P17861 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079602 0.84 ALDH1A1 (0.64) LMNAPKMHTTMEN1KMT2A
SCHEMBL10702111 0.82 LMNA (0.56) LMNAPKMHTTMEN1KMT2A
SCHEMBL7080668 0.81 MEN1 (0.54) LMNAPKMHTTMEN1KMT2A
SCHEMBL7075758 0.81 PKM (0.63) LMNAPKMHTTMEN1KMT2A
SCHEMBL20635988 0.80 SMN1; SMN2 (0.61) LMNAPKMHTTMEN1KMT2A
SCHEMBL7109414 0.80 LMNA (0.51) LMNAPKMHTTMEN1KMT2A
SCHEMBL7082412 0.79 LMNA (0.53) LMNAPKMHTTMEN1KMT2A
SCHEMBL7079622 0.76 HTR1A (0.55) LMNAPKMHTTMEN1KMT2A
SCHEMBL7075094 0.76 MEN1 (0.48) LMNAHTTMEN1KMT2AALDH1A1
SCHEMBL23052441 0.76 ALDH1A1 (0.64) PKMMEN1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030158186-A1 Compositions and methods for treating heart failure CYTOKINETICS, INCORPORATED 2003-08-21 US disclosed
WO-2003059265-A2 COMPOSITIONS AND METHODS FOR TREATING HEART FAILURE CYTOKINETICS, INC. (US) 2003-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030158186-A1 Compositions and methods for treating heart failure MYH2, TNNI3, MYLK2 LMNA 228/4885PKM 1445/4885HTT 3632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.