SCHEMBL7080668

SCHEMBL7080668

CC(O)c1ccc(S(=O)(=O)NC2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
LMNA P02545 1/20 0.53
MCOLN3 Q8TDD5 1/20 0.51
HTT P42858 2/20 0.50
ALDH1A1 P00352 2/20 0.50
POLB P06746 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
EPHX2 P34913 1/20 0.48
UCHL1 P09936 1/20 0.48
USP30 Q70CQ3 1/20 0.48
PKM P14618 2/20 0.47
CNR1 P21554 1/20 0.47
CCR6 P51684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082412 0.88 LMNA (0.53) MEN1KMT2ALMNAMCOLN3HTT
SCHEMBL7075094 0.85 MEN1 (0.48) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL7079602 0.84 ALDH1A1 (0.64) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL7075758 0.81 PKM (0.63) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL7080360 0.81 LMNA (0.52) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL10702111 0.80 LMNA (0.56) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL7109414 0.78 LMNA (0.51) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL7079622 0.76 HTR1A (0.55) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL23052441 0.74 ALDH1A1 (0.64) MEN1KMT2AALDH1A1POLBUCHL1
SCHEMBL14923992 0.73 USP30 (0.64) MEN1KMT2ALMNAMCOLN3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030158186-A1 Compositions and methods for treating heart failure CYTOKINETICS, INCORPORATED 2003-08-21 US disclosed
WO-2003059265-A2 COMPOSITIONS AND METHODS FOR TREATING HEART FAILURE CYTOKINETICS, INC. (US) 2003-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030158186-A1 Compositions and methods for treating heart failure MYH2, TNNI3, MYLK2 MEN1 4537/4885KMT2A 2747/4885LMNA 228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.