SCHEMBL7080948

SCHEMBL7080948

O=C(CCCN1CCN(c2ccc3ncccc3c2)CC1)c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.67
DRD4 P21917 9/20 0.67
HTR1A P08908 9/20 0.67
DRD3 P35462 9/20 0.67
HTR2A P28223 8/20 0.67
HTR2C P28335 6/20 0.67
HRH1 P35367 4/20 0.67
ADRA2C P18825 2/20 0.67
TMEM97 Q5BJF2 5/20 0.63
SIGMAR1 Q99720 5/20 0.63
HTR7 P34969 4/20 0.63
LMNA P02545 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2D6 P10635 1/20 0.63
CYP2C9 P11712 1/20 0.63
CYP2C19 P33261 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
CHRM1 P11229 1/20 0.57
DRD1 P21728 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083839 0.84 DRD2 (0.61) DRD2DRD4HTR1ADRD3HTR2A
SCHEMBL11832182 0.81 DRD2 (0.88) DRD2DRD4HTR1ADRD3HTR2A
SCHEMBL2027077 0.80 DRD2 (0.69) DRD2DRD4HTR1ADRD3HTR2A
SCHEMBL6234537 0.78 DRD2 (0.77) DRD2DRD4HTR1ADRD3HTR2A
Hydrochloric Acid SCHEMBL6708494 0.78 DRD2 (0.67) DRD2DRD4HTR1ADRD3HTR2A
Azaperone SCHEMBL29437229 0.78 DRD4 (1.00) DRD2DRD4HTR1ADRD3HTR2A
Azaperone SCHEMBL121134 0.78 DRD4 (1.00) DRD2DRD4HTR1ADRD3HTR2A
Cinuperone SCHEMBL31395265 0.76 HTR1A (0.70) DRD2DRD4HTR1ADRD3HTR2A
Cinuperone SCHEMBL678891 0.76 HTR1A (0.70) DRD2DRD4HTR1ADRD3HTR2A
SCHEMBL11833639 0.76 DRD2 (0.78) DRD2DRD4HTR1ADRD3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326842-A1 ARYLPIPERAZINE DERIVATIVES AND THEIR USE AS PSYCHOTROPIC AGENTS MERCK PATENT GmbH (DE) 2003-07-16 EP disclosed
WO-2002020491-A1 ARYLPIPERAZINE DERIVATIVES AND THEIR USE AS PSYCHOTROPIC AGENTS MERCK PATENT GMBH (DE) 2002-03-14 WO disclosed