SCHEMBL7081609

SCHEMBL7081609

c1ccc(N2CCN(CCc3nc4c(s3)CCc3ccccc3-4)CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.46
HTR1A P08908 5/20 0.46
ADORA1 P30542 1/20 0.45
DRD3 P35462 4/20 0.44
DRD4 P21917 2/20 0.44
KCNH2 Q12809 1/20 0.42
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
DRD5 P21918 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
HTR7 P34969 2/20 0.41
ADRB2 P07550 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
ADRB1 P08588 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
ATP4A P20648 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6957118 0.99 DRD2 (0.45) DRD2HTR1AADORA1DRD3DRD4
SCHEMBL6952045 0.93 DRD3 (0.53) DRD2HTR1AADORA1DRD3DRD4
Hydrochloric Acid SCHEMBL6960476 0.92 DRD3 (0.52) DRD2HTR1AADORA1DRD3DRD4
SCHEMBL6952207 0.92 HTR1A (0.49) DRD2HTR1ADRD3DRD4KCNH2
Hydrochloric Acid SCHEMBL6959796 0.91 HTR1A (0.48) DRD2HTR1ADRD3DRD4KCNH2
SCHEMBL6953511 0.88 ADORA1 (0.47) DRD2ADORA1DRD3DRD4HTR7
Hydrochloric Acid SCHEMBL6959246 0.87 ADORA1 (0.46) DRD2ADORA1DRD3DRD4HTR7
SCHEMBL7082241 0.79 SIGMAR1 (0.52) DRD2HTR1AADORA1DRD3DRD4
Hydrochloric Acid SCHEMBL6956636 0.78 DRD2 (0.52) DRD2HTR1AADORA1DRD3DRD4
SCHEMBL7084707 0.75 SIGMAR1 (0.57) DRD2HTR1ADRD3DRD4ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0851862-B1 1(HETERO)ARYL-4-(CONDENSED THIAZOL-2-YLALKYL)-PIPERAZINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF 5-HT1A-RECEPTOR MEDIATED DISORDERS PHARMACIA ITALIA SPA (IT) 2003-09-10 EP claimed