SCHEMBL7085833

SCHEMBL7085833

O=[N+]([O-])c1cc(Br)c(Oc2ccc3[nH]ccc3c2)c(Br)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.41
AHR P35869 1/20 0.41
NR4A2 P43354 1/20 0.41
THRA P10827 3/20 0.40
THRB P10828 3/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
JAK2 O60674 1/20 0.38
PRKCQ Q04759 2/20 0.38
MAOA P21397 1/20 0.38
HDAC1 Q13547 1/20 0.38
ALDH1A1 P00352 2/20 0.37
GLA P06280 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
NQO2 P16083 1/20 0.35
LTA4H P09960 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084821 0.84 THRA (0.53) THRATHRBPTGS1PTGS2JAK2
SCHEMBL22632403 0.84 THRA (0.51) AHRNR4A2THRATHRBPTGS1
SCHEMBL7088569 0.81 THRA (0.53) AHRTHRATHRBPTGS1PTGS2
SCHEMBL7091630 0.80 AHR (0.47) CYP2A6AHRNR4A2THRATHRB
SCHEMBL7089721 0.76 THRA (0.45) THRATHRBALDH1A1GLALTA4H
SCHEMBL3484001 0.74 PDE7A (0.59) ALDH1A1GLAMAPTHTT
SCHEMBL3053391 0.74 HSPB1 (0.56) ALDH1A1MAPTHTT
SCHEMBL2468340 0.74 CTSV (0.56) PTGS1PTGS2MAOAMAPTHTT
SCHEMBL29821791 0.74 ALDH1A1 (0.46) PTGS2ALDH1A1GLANQO2MAPT
SCHEMBL7090515 0.73 THRA (0.56) THRATHRBHDAC1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268422-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES Bayer Aktiengesellschaft (DE) 2003-01-02 EP disclosed
WO-2001070687-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-27 WO disclosed