SCHEMBL7086385

SCHEMBL7086385

CC(C)c1nc(COC(N)=O)n(Cc2cccnc2)c1Sc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 4/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
S1PR3 Q99500 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRA5 P31644 1/20 0.35
MDM2 Q00987 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
HIF1A Q16665 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960297 0.92 MDM2 (0.34) TLR7L3MBTL1S1PR3ALDH1A1KDM4E
SCHEMBL6969306 0.92 KMT2A (0.39) L3MBTL1S1PR3ALDH1A1KDM4ECYP3A4
SCHEMBL6974469 0.91 TLR7 (0.36) TLR7L3MBTL1S1PR3ALDH1A1KDM4E
SCHEMBL7078695 0.90 CYP1A2 (0.36) TLR7S1PR3ALDH1A1KDM4ECYP3A4
SCHEMBL6967707 0.90 ALDH1A1 (0.40) S1PR3ALDH1A1GABRA1GABRA5LMNA
SCHEMBL6972373 0.90 PIM1 (0.36) TLR7L3MBTL1ALDH1A1KDM4EKMT2A
SCHEMBL6971258 0.89 LMNA (0.40) TLR7L3MBTL1S1PR3LMNA
SCHEMBL6967126 0.89 GRIN1 (0.37) TLR7S1PR3
SCHEMBL6957033 0.89 ADRA1D (0.37) TLR7S1PR3ALDH1A1GABRA1GABRA5
SCHEMBL6964229 0.89 TOP2A (0.41) L3MBTL1S1PR3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed