SCHEMBL6974469

SCHEMBL6974469

CC(C)c1nc(CCOC(N)=O)n(Cc2cccnc2)c1Sc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
S1PR3 Q99500 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CHRNA7 P36544 1/20 0.34
ENPP2 Q13822 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRA5 P31644 1/20 0.34
MDM2 Q00987 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971258 0.95 LMNA (0.40) TLR7HDAC1HDAC8L3MBTL1S1PR3
SCHEMBL6960297 0.92 MDM2 (0.34) TLR7HDAC1HDAC8L3MBTL1S1PR3
SCHEMBL7084562 0.92 KDM4E (0.37) TLR7HDAC1HDAC8L3MBTL1S1PR3
SCHEMBL7086385 0.91 TLR7 (0.35) TLR7L3MBTL1S1PR3LMNAHTT
SCHEMBL6973955 0.91 ALDH1A1 (0.35) TLR7HDAC1HDAC8S1PR3LMNA
SCHEMBL7080841 0.90 GRIN1 (0.36) S1PR3LMNAKMT2AENPP2ALDH1A1
SCHEMBL6973316 0.90 ALDH1A1 (0.39) LMNAKMT2ASMN1; SMN2ALDH1A1GABRA1
SCHEMBL6968774 0.90 PIM1 (0.35) TLR7LMNAKMT2AENPP2HIF1A
SCHEMBL6966178 0.90 ADRA1D (0.36) S1PR3KMT2AALDH1A1GABRA1GABRA5
SCHEMBL6974966 0.90 GRIN1 (0.36) TLR7HDAC1HDAC8S1PR3ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed