SCHEMBL7092539

SCHEMBL7092539

Nc1ccccc1Cn1cc(-c2ccco2)cn1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.50
ADORA1 P30542 7/20 0.50
ADORA3 P0DMS8 3/20 0.45
ADORA2B P29275 3/20 0.45
SCD5 Q86SK9 7/20 0.43
SCD O00767 3/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
TAAR1 Q96RJ0 1/20 0.38
CREBBP Q92793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6693877 0.84 ALDH1A1 (0.56) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL7004006 0.80 L3MBTL1 (0.64) ADORA2AADORA1SCD5SCDALDH1A1
SCHEMBL7097845 0.79 ADORA2A (0.43) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL7096885 0.76 ADORA2A (0.52) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL3549869 0.76 HDAC1 (0.61) ADORA2AADORA1ADORA2BSCD5ALDH1A1
SCHEMBL7094550 0.75 DAO (0.39) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL6691423 0.75 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL7092817 0.75 SCD5 (0.45) ADORA2AADORA1ADORA3ADORA2BSCD5
SCHEMBL8357391 0.74 PIM1 (0.45) ADORA2AADORA1SCD5SCDALDH1A1
SCHEMBL7091724 0.73 ADORA2A (0.45) ADORA2AADORA1ALDH1A1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed