SCHEMBL7097845

SCHEMBL7097845

c1coc(Cn2cc(-c3ccco3)cn2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.43
ADORA1 P30542 2/20 0.43
ALDH1A1 P00352 4/20 0.43
TSHR P16473 4/20 0.43
HSD17B10 Q99714 3/20 0.43
KDM4E B2RXH2 3/20 0.43
USP2 O75604 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 2/20 0.40
MAPT P10636 2/20 0.40
NPC1 O15118 1/20 0.40
MITF O75030 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004006 0.83 L3MBTL1 (0.64) ADORA2AADORA1ALDH1A1TSHRHSD17B10
SCHEMBL6691423 0.81 ADORA2A (0.48) ADORA2AADORA1ALDH1A1TSHRKDM4E
SCHEMBL7098488 0.79 L3MBTL1 (0.57) ADORA2AADORA1ALDH1A1HSD17B10KDM4E
SCHEMBL7092539 0.79 ADORA2A (0.50) ADORA2AADORA1ALDH1A1L3MBTL1POLB
SCHEMBL6693877 0.79 ALDH1A1 (0.56) ADORA2AADORA1ALDH1A1KDM4EL3MBTL1
SCHEMBL7096885 0.76 ADORA2A (0.52) ADORA2AADORA1L3MBTL1MEN1KMT2A
SCHEMBL6690784 0.76 ADORA2A (0.50) ADORA2AADORA1ALDH1A1KDM4EL3MBTL1
SCHEMBL6693887 0.74 MEN1 (0.60) ADORA2AADORA1ALDH1A1TSHRHSD17B10
SCHEMBL7094550 0.73 DAO (0.39) ADORA2AADORA1ALDH1A1L3MBTL1POLB
SCHEMBL7093005 0.73 SCD5 (0.55) ADORA2AADORA1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed