SCHEMBL7093597

SCHEMBL7093597

COc1ccc(CNC(=O)c2ccnc(C(=O)OC(N)c3ccc(OC)cc3OC)c2)c(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
TSHR P16473 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
MAPT P10636 2/20 0.48
HPGD P15428 3/20 0.46
GAA P10253 2/20 0.46
ROCK2 O75116 1/20 0.46
TP53 P04637 4/20 0.46
LMNA P02545 4/20 0.46
ABCB1 P08183 1/20 0.46
NAMPT P43490 1/20 0.45
TAS1R3 Q7RTX0 2/20 0.45
TAS1R1 Q7RTX1 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
PKM P14618 1/20 0.43
HTT P42858 1/20 0.43
MAOB P27338 1/20 0.43
PPARG P37231 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212964 0.86 ALDH1A1 (0.65) ALDH1A1TSHRNPSR1MAPTHPGD
SCHEMBL6258412 0.79 ROCK2 (0.55) MAPTHPGDGAAROCK2TP53
SCHEMBL6255361 0.76 WDR5 (0.48) MAPTROCK2TP53LMNANAMPT
SCHEMBL7142998 0.75 MEN1 (0.43) MAOBPPARG
SCHEMBL22774462 0.75 POLB (0.62) ALDH1A1MAPTHPGDGAAROCK2
SCHEMBL29453012 0.75 POLB (0.62) ALDH1A1MAPTHPGDGAAROCK2
SCHEMBL6258517 0.74 ROS1 (0.48) ALDH1A1MAPTLMNANAMPT
SCHEMBL5329065 0.74 LMNA (0.60) ALDH1A1TSHRNPSR1MAPTHPGD
SCHEMBL23985268 0.74 ALDH1A1 (0.64) ALDH1A1TSHRNPSR1MAPTHPGD
SCHEMBL30305464 0.74 ALDH1A1 (0.64) ALDH1A1TSHRNPSR1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362033-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP claimed
WO-2002064568-A1 PYRIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed