SCHEMBL7094551

SCHEMBL7094551

CS(=O)(=O)Nc1cccc(N(c2ccccc2)C(CN)c2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.56
NR3C2 P08235 4/20 0.48
HTR7 P34969 2/20 0.47
KEAP1 Q14145 1/20 0.46
ALDH1A1 P00352 2/20 0.44
ADRA2C P18825 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
MAPKAPK2 P49137 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093212 0.96 NR3C1 (0.54) NR3C1NR3C2HTR7KEAP1ALDH1A1
SCHEMBL7094983 0.89 NR3C2 (0.57) NR3C1NR3C2KEAP1ALDH1A1SMN1; SMN2
SCHEMBL7094549 0.78 NR3C1 (0.52) NR3C1NR3C2HTR7KEAP1ALDH1A1
SCHEMBL7093211 0.76 NR3C1 (0.50) NR3C1NR3C2HTR7KEAP1ALDH1A1
SCHEMBL7093914 0.76 TAAR1 (0.52) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL7094120 0.75 SLC6A2 (0.41) CYP3A4
SCHEMBL11420225 0.75 ADRB3 (0.61) KEAP1ALDH1A1ADRA2CADRA1AADRA1B
SCHEMBL9481726 0.74 NR3C2 (0.78) NR3C1NR3C2HTR7KEAP1ALDH1A1
SCHEMBL11570895 0.74 ALDH1A1 (0.50) NR3C1KEAP1ALDH1A1ADRA2CADRA1A
SCHEMBL4370199 0.74 KEAP1 (0.52) NR3C1KEAP1ALDH1A1SMN1; SMN2MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082777-A2 NOVEL GLUCOCORTICOID RECEPTOR LIGANDS KARO BIO AB (SE) 2003-10-09 WO claimed
WO-2003082777-A2 NOVEL GLUCOCORTICOID RECEPTOR LIGANDS KARO BIO AB (SE) 2003-10-09 WO disclosed