SCHEMBL7108875

SCHEMBL7108875

O=C(NCC(O)CO)c1cncc(C(=O)[N+](CC(O)CO)(CC(O)CO)CC(O)CO)n1.O=C(c1cnc(C(=O)N(CC(O)CO)CC(O)CO)cn1)N(CC(O)CO)CC(O)CO

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.31
HIF1A Q16665 1/20 0.31
ICAM1 P05362 1/20 0.31
SELE P16581 1/20 0.31
CNR2 P34972 1/20 0.31
ROCK2 O75116 1/20 0.31
MAP2K1 Q02750 2/20 0.30
SMO Q99835 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7109193 0.79 ICAM1 (0.40) ICAM1SELECNR2MAP2K1SMO
SCHEMBL7108469 0.76 CNR2 (0.41) CYP2C19HIF1AICAM1SELECNR2
SCHEMBL7107198 0.73
SCHEMBL7106667 0.73 KCNA5 (0.31)
SCHEMBL7105165 0.71 MAP2K1 (0.41) CYP2C19HIF1AICAM1SELECNR2
SCHEMBL7110604 0.70 LMNA (0.41) CYP2C19HIF1AICAM1SELECNR2
SCHEMBL7104658 0.68 SMN1; SMN2 (0.35) CYP2C19
SCHEMBL590665 0.68 SIRT6 (0.42)
SCHEMBL18230701 0.65 SIRT6 (0.42) ICAM1SELECNR2MAP2K1SMO
SCHEMBL28237026 0.65 SMN1; SMN2 (0.54) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001944-B1 PYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA SA (FR) 2003-10-01 EP claimed