SCHEMBL7109213

SCHEMBL7109213

CC(=O)OC1Cc2ccc([N+](=O)[O-])cc2C1N(OC(C)(C)C)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
MAPT P10636 3/20 0.34
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
DRD2 P14416 1/20 0.33
PNMT P11086 4/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
AR P10275 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
NR3C2 P08235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7101387 0.85 CHRNB2 (0.37) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL7101254 0.77 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19CHRNB2CHRNB4
SCHEMBL7101251 0.77 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19CHRNB2CHRNB4
SCHEMBL7149109 0.69 ALDH1A1 (0.41) CYP3A4CYP2C9CYP2C19CHRNB2CHRNB4
SCHEMBL7149107 0.69 ALDH1A1 (0.41) CYP3A4CYP2C9CYP2C19CHRNB2CHRNB4
SCHEMBL7107511 0.67 KDM4E (0.45) MAPTALDH1A1KDM4ELMNA
SCHEMBL7107514 0.67 KDM4E (0.45) MAPTALDH1A1KDM4ELMNA
SCHEMBL6988386 0.67 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19ALDH1A1DRD2
SCHEMBL7149111 0.67 GAA (0.43) MAPTALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL8308233 0.67 CHRM4 (0.47) CYP3A4CYP2C9CYP2C19MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923543-B1 POTASSIUM CHANNEL INHIBITORS ICAGEN INC (US) 2003-09-24 EP disclosed
US-6083986-A Potassium channel inhibitors ICAGEN, INC. (US) 2000-07-04 US disclosed