SCHEMBL7121887

SCHEMBL7121887

CC(C)(C)OC(=O)NCC1CN(C(=O)OC(C)(C)C)CCC1N(CC(=O)O)C(=O)c1ccccc1.NC(=O)c1ccc2c(c1)CCC2

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
USP30 Q70CQ3 2/20 0.40
GPR119 Q8TDV5 4/20 0.39
NOD2 Q9HC29 1/20 0.38
NOD1 Q9Y239 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
KDM1A O60341 2/20 0.38
DRD2 P14416 1/20 0.36
LIMK2 P53671 1/20 0.35
PARP14 Q460N5 1/20 0.35
CHEK2 O96017 2/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4812628 0.80 GPR119 (0.42) NPC1RAB9AKDM4EPKMUSP30
SCHEMBL7121817 0.73 HSD17B3 (0.41) LIMK2
SCHEMBL7429016 0.71 NPC1 (0.35) NPC1RAB9AKDM4EMEN1KMT2A
Trifluoroacetic Acid SCHEMBL7433732 0.70 SLC6A2 (0.34)
SCHEMBL7430527 0.70 PDK1 (0.34) NPC1RAB9AKDM4EMEN1KMT2A
SCHEMBL7430920 0.69 PDK1 (0.34) NPC1RAB9AMEN1KMT2A
SCHEMBL5210913 0.68 NPC1 (0.39) NPC1RAB9AKDM4E
SCHEMBL5210889 0.67 NPC1 (0.40) NPC1RAB9AKDM4E
SCHEMBL5216930 0.67 RAB9A (0.37) NPC1RAB9AKDM4E
SCHEMBL5210074 0.67 RXRB (0.38) NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294691-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2003-03-26 EP disclosed
WO-2001096305-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2001-12-20 WO disclosed