SCHEMBL7122553

SCHEMBL7122553

CCN(c1cccc(Br)c1)S(=O)(=O)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.43
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA5A P35218 1/20 0.40
CA9 Q16790 1/20 0.40
TSHR P16473 3/20 0.37
MAPK1 P28482 2/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
LMNA P02545 3/20 0.37
KDM4E B2RXH2 1/20 0.37
RECQL P46063 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTT P42858 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14855516 0.81 L3MBTL1 (0.47) CA1CA2CA5ACA9LMNA
SCHEMBL7117168 0.81 NR1I2 (0.40) RORCCA1CA2CA5ACA9
SCHEMBL7128846 0.80 CA1 (0.42) CA1CA2CA5ACA9TSHR
SCHEMBL19065098 0.77 HDAC8 (0.64) RORCTSHRKMT2AHDAC3HDAC11
SCHEMBL6624409 0.74 ESR1 (0.52) RORCCA9TSHRMAPK1KMT2A
SCHEMBL7896008 0.73 ALDH1A1 (0.59) TSHRMAPK1KMT2ALMNAKDM4E
SCHEMBL14855515 0.70 CA1 (0.37) CA1CA2CA5ACA9KMT2A
SCHEMBL5731154 0.68 RORC (0.57) RORCKMT2AALDH1A1SMN1; SMN2ESR1
SCHEMBL3818736 0.68 ALDH1A1 (0.41) TSHRMAPK1LMNAALDH1A1CYP3A4
SCHEMBL4064736 0.68 HTR7 (0.44) TSHRMAPK1LMNAALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed