SCHEMBL7128846

SCHEMBL7128846

CN(c1cccc(Br)c1)S(=O)(=O)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
NR1H3 Q13133 2/20 0.40
HSD17B1 P14061 3/20 0.38
HSD17B2 P37059 3/20 0.38
SIRT2 Q8IXJ6 1/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
GBA1 P04062 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7119808 0.80 KIF11 (0.42) CA1CA2CA5ACA9NR1H3
SCHEMBL7122553 0.80 RORC (0.43) CA1CA2CA5ACA9TSHR
SCHEMBL2634503 0.79 ALDH1A1 (0.50) HTTL3MBTL1ALDH1A1MAPK1
SCHEMBL9888504 0.78 NR1H3 (0.49) CA2CA9NR1H3HTTALDH1A1
SCHEMBL14855515 0.73 CA1 (0.37) CA1CA2CA5ACA9L3MBTL1
SCHEMBL14855516 0.73 L3MBTL1 (0.47) CA1CA2CA5ACA9HTT
SCHEMBL31349768 0.72 ALDH1A1 (0.31) ALDH1A1
SCHEMBL27720036 0.70 ALDH1A1 (0.44) TSHRL3MBTL1MTNR1AMTNR1BALDH1A1
SCHEMBL7983296 0.70 RIPK1 (0.41) CA1CA2CA5ACA9HSD17B1
SCHEMBL21594681 0.69 ALDH1A1 (0.48) MTNR1AMTNR1BALDH1A1MAPK1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed