SCHEMBL7124501

SCHEMBL7124501

CNC(=O)c1ccc(S(=O)(=O)NC(CCc2ccccc2)C(=O)NC(C)(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.54
HPN P05981 1/20 0.54
MMP3 P08254 1/20 0.49
MMP9 P14780 4/20 0.49
PSMB8 P28062 4/20 0.49
PSMB5 P28074 4/20 0.49
MMP2 P08253 2/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPT P10636 1/20 0.49
MEN1 O00255 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
KMT2A Q03164 1/20 0.48
USP30 Q70CQ3 2/20 0.46
MMP7 P09237 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ITGB3 P05106 2/20 0.45
ITGA2B P08514 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7124459 0.89 ALDH1A1 (0.57) PLAUHPNMMP9PSMB8PSMB5
SCHEMBL7127019 0.88 PLAU (0.60) PLAUHPNMMP9PSMB8PSMB5
SCHEMBL7127817 0.87 MMP2 (0.53) PLAUHPNMMP9PSMB8PSMB5
SCHEMBL7117861 0.86 PSMB8 (0.54) PLAUHPNMMP9PSMB8PSMB5
SCHEMBL7118677 0.85 MMP2 (0.49) PLAUHPNMMP9PSMB8PSMB5
SCHEMBL7116828 0.84 USP30 (0.43) PLAUHPNMMP3MMP9PSMB8
SCHEMBL7121669 0.84 ALDH1A1 (0.63) PLAUHPNMMP3MMP9MMP2
SCHEMBL7127030 0.84 PSMB8 (0.51) PLAUHPNMMP3MMP9PSMB8
SCHEMBL7118405 0.83 MMP2 (0.50) PLAUHPNMMP3MMP9PSMB8
SCHEMBL7125293 0.83 PLAU (0.59) PLAUHPNMMP9PSMB8MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583318-B2 Carrying out a four component condensation reaction between components consisting of a sulfonamide, an aldehyde or ketone, an isocyanide and a carboxylic acid, and one of such components being attached to a solid support ADVANCED SYNTECH, LLC 2003-06-24 US disclosed
US-20030013910-A1 Method for synthesis of alpha-sulfonamido amide, carboxylic acid and hydroxamic acid derivatives ADVANCED SYNTECH LLC 2003-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030013910-A1 Method for synthesis of alpha-sulfonamido amide, carboxylic acid and hydroxamic acid derivatives ASPH, COASY, HAAO PLAU 1115/4885HPN 247/4885MMP3 2528/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.