SCHEMBL7127619

SCHEMBL7127619

O=C1CC(NC2Cc3ccccc3C2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
ACHE P22303 2/20 0.40
CYP19A1 P11511 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
SIGMAR1 Q99720 1/20 0.36
S100A4 P26447 1/20 0.36
BCHE P06276 2/20 0.35
CES1 P23141 1/20 0.35
HTR7 P34969 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
AR P10275 1/20 0.35
HSD11B1 P28845 1/20 0.35
AKR1C3 P42330 1/20 0.35
CYP2A6 P11509 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7120126 0.98 P2RX7 (0.39) P2RX7ACHECYP19A1CA1CA2
SCHEMBL6863573 0.83 BCHE (0.53) P2RX7ACHES100A4BCHEALDH1A1
Hydrochloric Acid SCHEMBL6863833 0.82 BCHE (0.51) P2RX7ACHES100A4BCHEALDH1A1
SCHEMBL3702992 0.82 BCHE (0.56) P2RX7ACHEBCHEALDH1A1
SCHEMBL7126444 0.80 MAOA (0.51) P2RX7ACHECA1CA2BCHE
Hydrochloric Acid SCHEMBL7117163 0.78 MAOA (0.50) P2RX7ACHECA1CA2BCHE
SCHEMBL18988275 0.75 S100A4 (0.44) P2RX7CYP19A1S100A4ALDH1A1ADORA3
SCHEMBL29908700 0.75 S100A4 (0.44) P2RX7CYP19A1S100A4ALDH1A1ADORA3
SCHEMBL2404815 0.75 SLC6A2 (0.44) P2RX7S100A4ADORA3ARHSD11B1
SCHEMBL6589968 0.71 CA1 (0.52) CA1CA2SIGMAR1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874800-B1 INDANE DIMER COMPOUNDS WITH SMOOTH MUSCLE RELAXING AND/OR MAST CELL STABILISING AND/OR ANTIINFLAMMATORY ACTIVITY VENANTIUS LTD (IE) 2003-08-06 EP claimed
US-6423752-B1 SUCH AS 3-(N-1-INDANYLAMINO)-INDAN-1-ONE 3-(N-1-INDANYLAMINO) INDAN-1-ONE FORMED BY REACTING AMINO-INDANE COMPOUND WITH BROMO-INDANONE COMPOUND IN PRESENCE OF TRIETHYLENEAMINE VENANTIUS LIMITED (IE) 2002-07-23 US claimed
US-20020052530-A1 INDANE DIMER COMPOUNDS WITH SMOOTH MUSCLE RELAXING AND/OR MAST CELL STABILISING AND/OR ANTIINFLAMMATORY ACTIVITY VENANTIUS LIMITED (IE) 2002-05-02 US claimed
EP-0874800-B1 INDANE DIMER COMPOUNDS WITH SMOOTH MUSCLE RELAXING AND/OR MAST CELL STABILISING AND/OR ANTIINFLAMMATORY ACTIVITY VENANTIUS LTD (IE) 2003-08-06 EP disclosed
US-6423752-B1 SUCH AS 3-(N-1-INDANYLAMINO)-INDAN-1-ONE 3-(N-1-INDANYLAMINO) INDAN-1-ONE FORMED BY REACTING AMINO-INDANE COMPOUND WITH BROMO-INDANONE COMPOUND IN PRESENCE OF TRIETHYLENEAMINE VENANTIUS LIMITED (IE) 2002-07-23 US disclosed
WO-1997020805-A1 INDANE DIMER COMPOUNDS WITH SMOOTH MUSCLE RELAXING AND/OR MAST CELL STABILISING AND/OR ANTIINFLAMMATORY ACTIVITY VENANTIUS LIMITED (IE) 1997-06-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020052530-A1 INDANE DIMER COMPOUNDS WITH SMOOTH MUSCLE RELAXING AND/OR MAST CELL STABILISING AND/OR ANTIINFLAMMATORY ACTIVITY MYLK, HRH2, HRH1 P2RX7 1149/4885ACHE 861/4885CYP19A1 1657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.