SCHEMBL7130522

SCHEMBL7130522

Cc1ccc(Oc2cccc(C=C3C(=O)Nc4ccc(Br)c(C)c43)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 5/20 0.51
MEN1 O00255 5/20 0.50
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
KMT2A Q03164 5/20 0.50
POLB P06746 3/20 0.50
NTRK1 P04629 1/20 0.46
TDP1 Q9NUW8 2/20 0.43
ATM Q13315 1/20 0.41
AKR1B1 P15121 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
LRRK2 Q5S007 1/20 0.40
KDM1A O60341 1/20 0.40
MMP3 P08254 1/20 0.39
MMP13 P45452 1/20 0.39
RET P07949 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7133306 0.93 ADAMTS5 (0.50) ADAMTS5MEN1NPC1RAB9AKMT2A
SCHEMBL7136320 0.90 ADAMTS5 (0.54) ADAMTS5MEN1NPC1RAB9AKMT2A
SCHEMBL7137562 0.89 ADAMTS5 (0.52) ADAMTS5MEN1NPC1RAB9AKMT2A
SCHEMBL7134866 0.87 LRRK2 (0.50) MEN1NPC1RAB9AKMT2APOLB
SCHEMBL7140874 0.86 ADAMTS5 (0.43) ADAMTS5MEN1NPC1RAB9AKMT2A
SCHEMBL7136206 0.85 RET (0.50) KMT2APOLBNTRK1AKR1B1L3MBTL1
SCHEMBL7136012 0.85 ADAMTS5 (0.51) ADAMTS5MEN1NPC1RAB9AKMT2A
SCHEMBL7134014 0.81 RET (0.48) MEN1NPC1RAB9AKMT2APOLB
SCHEMBL7134020 0.81 LRRK2 (0.49) MAOAMAOBLRRK2RET
SCHEMBL7135594 0.81 MMP13 (0.50) ADAMTS5MEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed