SCHEMBL7133306

SCHEMBL7133306

COc1ccc(Oc2cccc(C=C3C(=O)Nc4ccc(Br)c(C)c43)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 3/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
POLB P06746 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
LRRK2 Q5S007 1/20 0.46
NTRK1 P04629 1/20 0.45
RET P07949 2/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
PIM1 P11309 2/20 0.41
AKR1B1 P15121 2/20 0.41
METAP1 P53582 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
MDM2 Q00987 1/20 0.41
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7130522 0.93 ADAMTS5 (0.51) ADAMTS5MEN1KMT2ANPC1RAB9A
SCHEMBL7134866 0.92 LRRK2 (0.50) MEN1KMT2ANPC1RAB9APOLB
SCHEMBL7136320 0.89 ADAMTS5 (0.54) ADAMTS5MEN1KMT2ANPC1RAB9A
SCHEMBL7137562 0.88 ADAMTS5 (0.52) ADAMTS5MEN1KMT2ANPC1RAB9A
SCHEMBL7132312 0.85 ADAMTS5 (0.50) ADAMTS5MEN1KMT2ANPC1RAB9A
SCHEMBL7140874 0.85 ADAMTS5 (0.43) ADAMTS5MEN1KMT2ANPC1RAB9A
SCHEMBL7136206 0.85 RET (0.50) KMT2APOLBL3MBTL1LRRK2NTRK1
SCHEMBL7134020 0.80 LRRK2 (0.49) LRRK2RETPIM1PIM2MDM2
SCHEMBL7135594 0.80 MMP13 (0.50) ADAMTS5MEN1KMT2ANPC1RAB9A
SCHEMBL7136994 0.79 MAOA (0.44) MEN1KMT2ARETPIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed