SCHEMBL714053

SCHEMBL714053

CC1(C)OCC(CC[O])O1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.49
ALDH1A1 P00352 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TMEM97 Q5BJF2 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM3 P20309 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7154999 0.86 CA2 (0.50) CA2ALDH1A1NPSR1TMEM97SIGMAR1
SCHEMBL18817541 0.86 CA2 (0.50) CA2ALDH1A1NPSR1TMEM97SIGMAR1
SCHEMBL717188 0.86 CA2 (0.45) CA2ALDH1A1NPSR1TMEM97SIGMAR1
SCHEMBL1526302 0.84 CA2 (0.46) CA2ALDH1A1NPSR1TMEM97SIGMAR1
SCHEMBL4475938 0.84 CA2 (0.46) CA2ALDH1A1NPSR1TMEM97SIGMAR1
SCHEMBL1526299 0.84 CA2 (0.46) CA2ALDH1A1NPSR1TMEM97SIGMAR1
SCHEMBL589481 0.82
SCHEMBL4421192 0.82
SCHEMBL589285 0.82
SCHEMBL13130046 0.82 CA2 (0.47) CA2ALDH1A1NPSR1TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8324378-B2 Prodrugs and conjugates of prenylation inhibitors PURDUE RESEARCH FOUNDATION (US) 2012-12-04 US disclosed
US-8268959-B2 Suitable for binding high explosives, and may also be used as explosives in their own right; materials possess high energy density and are highly amenable to chemical modification thereby allowing for modification to the physical properties of the material; tacky and rubbery nature THE SECRETARY OF STATE FOR DEFENSE (GB) 2012-09-18 US disclosed
EP-2460842-A2 Novel energetic polyphosphazenes The Secretary of State For Defence (GB) 2012-06-06 EP disclosed
US-20120053356-A1 NOVEL ENERGETIC POLYPHOSPHAZENES THE SECRETARY OF STATE FOR DEFENSE (GB) 2012-03-01 US disclosed
US-20100249072-A1 PRODRUGS AND CONJUGATES OF PRENYLATION INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2010-09-30 US disclosed
WO-2009029849-A1 PRODRUGS AND CONJUGATES OF PRENYLATION INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2009-03-05 WO disclosed
EP-1960456-A1 NOVEL ENERGETIC POLYPHOSPHAZENES THE SECRETARY OF STATE FOR DEFENCE (GB) 2008-08-27 EP disclosed
US-20080108784-A1 Suitable for binding high explosives, and may also be used as explosives in their own right; materials possess high energy density and are highly amenable to chemical modification thereby allowing for modification to the physical properties of the material; tacky and rubbery nature DEFENSE, THE SECRETARY OF THE STATE FOR (GB) 2008-05-08 US disclosed
WO-2006099313-A2 PHOSPHATE CONJUGATES OF PRENYLATION INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2006-09-21 WO disclosed
WO-2006032882-A1 NOVEL ENERGETIC POLYPHOSPHAZENES THE SECRETARY OF STATE FOR DEFENCE (GB) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100249072-A1 PRODRUGS AND CONJUGATES OF PRENYLATION INHIBITORS FNTA, FNTB, FDPS CA2 1525/4885ALDH1A1 2414/4885NPSR1 3399/4885
US-20120053356-A1 NOVEL ENERGETIC POLYPHOSPHAZENES ACLY, PEBP1, DDX42 CA2 2462/4885ALDH1A1 4205/4885NPSR1 3269/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.