SCHEMBL7145016

SCHEMBL7145016

COc1cc(F)c2nccc(NC(=O)c3ncc[nH]3)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.40
GSK3B P49841 2/20 0.40
CDK5 Q00535 2/20 0.40
CDK8 P49336 1/20 0.40
CDK9 P50750 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
HDAC1 Q13547 2/20 0.40
BRAF P15056 1/20 0.40
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.37
KDR P35968 3/20 0.37
CLK2 P49760 2/20 0.37
HIPK4 Q8NE63 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37
MAP3K20 Q9NYL2 2/20 0.37
STK17A Q9UEE5 2/20 0.37
IRAK1 P51617 1/20 0.37
NEK4 P51957 1/20 0.37
MAP4K2 Q12851 1/20 0.37
SRPK1 Q96SB4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985604 0.81 HTR1A (0.51) GSK3AGSK3BCDK5HDAC1BRAF
SCHEMBL4277304 0.73 GSK3A (0.42) GSK3AGSK3BCDK5CDK8CDK9
SCHEMBL2817711 0.69 RAB9A (0.55) KMT2AMEN1RAB9ANPC1SMN1; SMN2
SCHEMBL2923376 0.69 NOS3 (0.40) KMT2AMEN1MAPK1RAB9ANPC1
SCHEMBL18544288 0.69 CCR1 (0.38) KMT2AMEN1DYRK1A
SCHEMBL30973172 0.69 MAP2K1 (0.42) GAAFPR2
SCHEMBL27588449 0.69 KDM4E (0.60) KDRAURKBAURKAMET
Oxalic Acid SCHEMBL5264185 0.68 LMNA (0.41) HDAC1KMT2AMEN1MAPK1PRKAA1
SCHEMBL3375901 0.66 CCR1 (0.38) KMT2AMEN1KDR
SCHEMBL4279169 0.66 NOS3 (0.43) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305308-A1 AMINOPIPERIDINE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2003-05-02 EP disclosed
WO-2002008224-A1 AMINOPIPERIDINE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY SMITHKLINE BEECHAM P.L.C. (GB) 2002-01-31 WO disclosed