SCHEMBL7146465

SCHEMBL7146465

CCOC(=O)c1cnc(NCCc2ccccn2)nc1-c1cccc([N+](=O)[O-])c1.CCOC(=O)c1cnc(NCCc2ccccn2)nc1-c1ccco1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.41
PDE4D Q08499 1/20 0.41
FOS P01100 1/20 0.41
JUN P05412 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
MAPT P10636 6/20 0.40
ALDH1A1 P00352 4/20 0.40
ADORA3 P0DMS8 7/20 0.38
ADORA2A P29274 7/20 0.38
ADORA1 P30542 7/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ADORA2B P29275 2/20 0.38
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5091586 0.93 FOS (0.46) PDE4APDE4DFOSJUNNFKB1
SCHEMBL5093408 0.88 ADORA3 (0.47) MAPTALDH1A1ADORA3ADORA2AADORA1
SCHEMBL7853285 0.88 FOS (0.44) FOSJUNNFKB1NFKB2RELA
SCHEMBL5092765 0.82 FOS (0.47) PDE4APDE4DFOSJUNNFKB1
SCHEMBL27570893 0.81 ALDH1A1 (0.46) PDE4APDE4DMAPTALDH1A1LMNA
SCHEMBL5098932 0.77 FOS (0.47) PDE4APDE4DFOSJUNNFKB1
SCHEMBL27559848 0.76 PKM (0.44) MAPTALDH1A1ADORA3ADORA2AADORA1
SCHEMBL5089195 0.76 ALDH1A1 (0.48) FOSJUNNFKB1NFKB2RELA
SCHEMBL5089370 0.75 MAPT (0.44) MAPTALDH1A1ADORA3ADORA2AADORA1
SCHEMBL5093430 0.75 RAB9A (0.49) MAPTALDH1A1LMNAMAPK1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed