SCHEMBL7149943

SCHEMBL7149943

CCSc1nc(C)c(CCO)c(=O)[nH]1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
PKM P14618 1/20 0.51
MCL1 Q07820 1/20 0.49
HPGD P15428 2/20 0.48
TSHR P16473 2/20 0.47
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.44
GLA P06280 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089906 0.84 PKM (0.55) ALDH1A1SMN1; SMN2PKMMCL1HPGD
SCHEMBL5108684 0.84 KDM4E (0.58) ALDH1A1PKMHPGDKDM4ELMNA
SCHEMBL7147721 0.76 GAA (0.46) ALDH1A1SMN1; SMN2PKMKDM4E
SCHEMBL10600602 0.76 PKM (0.49) ALDH1A1PKMHPGDTSHRKDM4E
SCHEMBL12143535 0.76 L3MBTL1 (0.46) ALDH1A1SMN1; SMN2TSHRKDM4ELMNA
SCHEMBL12142140 0.74 ALDH1A1 (0.40) ALDH1A1PKMHPGDKDM4E
SCHEMBL1895259 0.74 LMNA (0.74) ALDH1A1SMN1; SMN2HPGDTSHRLMNA
SCHEMBL512553 0.73 NPSR1 (0.58) ALDH1A1PKMKDM4E
SCHEMBL7146938 0.73 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2PKMKDM4ELMNA
SCHEMBL8515731 0.72 KDM4E (0.60) ALDH1A1PKMMCL1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2241567-A1 BICYCLOAMINE DERIVATIVE Eisai R&D Management Co., Ltd. (JP) 2010-10-20 EP disclosed
EP-0808313-B1 ANTIPSYCHOTIC 4-(1H-INDOLYL-1-YL)-1-SUBSTITUTED PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2003-08-13 EP disclosed
US-5919788-A PSYCHOLOGICAL DISORDERS JANSSEN PHARMACEUTICA, N.V. (BE) 1999-07-06 US disclosed
EP-0808313-A1 ANTIPSYCHOTIC 4-(1H-INDOLYL-1-YL)-1-SUBSTITUTED PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1997-11-26 EP disclosed
WO-1996023784-A1 ANTIPSYCHOTIC 4-(1H-INDOLYL-1-YL)-1-SUBSTITUTED PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1996-08-08 WO disclosed