SCHEMBL7150847

SCHEMBL7150847

COc1cccc(C(C=NO)c2cccc(Cl)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.39
AOC3 Q16853 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
MAPT P10636 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
CASR P41180 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PFKFB3 Q16875 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141858 0.87 NFE2L2 (0.39) NFE2L2L3MBTL1KDM4EKMT2AMAPT
SCHEMBL7094473 0.83 NFE2L2 (0.43) NFE2L2AOC3L3MBTL1KMT2ACHRM2
SCHEMBL7097655 0.69 NFE2L2 (0.44) NFE2L2L3MBTL1KDM4EKMT2AMAPT
SCHEMBL11619720 0.64 CASR (0.53) AOC3L3MBTL1CASR
SCHEMBL10954259 0.64 NFE2L2 (0.43) NFE2L2L3MBTL1KDM4EKMT2AMAPT
SCHEMBL11353744 0.64 AOC3 (0.45) AOC3L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL28031817 0.63 AOC3 (0.56) AOC3L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL17858535 0.63 DYRK1A (0.42) NFE2L2CASRSMN1; SMN2NPC1RAB9A
SCHEMBL2087869 0.63 AOC3 (0.59) AOC3L3MBTL1CHRM2CHRM1CHRM3
SCHEMBL2093768 0.63 AOC3 (0.59) AOC3L3MBTL1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366048-A2 PYRAZOLOPYRIDINE DERIVATIVES SmithKline Beecham Corporation (US) 2003-12-03 EP disclosed
WO-2002072581-A2 PYRAZOLOPYRIADINE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 2002-09-19 WO disclosed