SCHEMBL7154018

SCHEMBL7154018

N#Cc1ccc(NNC(=O)Oc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.46
MAPT P10636 5/20 0.45
KMT2A Q03164 5/20 0.45
ALDH1A1 P00352 5/20 0.45
MEN1 O00255 4/20 0.45
KDM4E B2RXH2 3/20 0.45
RAB9A P51151 2/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 1/20 0.45
PKM P14618 1/20 0.45
MAPK1 P28482 1/20 0.45
IL18 Q14116 1/20 0.45
RAD51 Q06609 1/20 0.44
GAA P10253 3/20 0.44
USP2 O75604 1/20 0.44
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
PLAU P00749 1/20 0.43
KLKB1 P03952 1/20 0.43
PRSS1 P07477 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10393667 0.84 ALDH1A1 (0.64) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL9553582 0.84 GAA (0.58) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL27802288 0.80 FAAH (0.51) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL1504425 0.80 PTGS2 (0.58) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL27785451 0.79 CHEK1 (0.45) MAPTKMT2AALDH1A1MEN1KDM4E
4-Cyanophenyl Phenylcarbamate SCHEMBL10393666 0.78 ALDH1A1 (0.64) MGLLMAPTKMT2AALDH1A1MEN1
SCHEMBL14108086 0.78 PTGS2 (0.65) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL20389099 0.77 MEN1 (0.61) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL28109363 0.76 LMNA (0.49) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL20379437 0.76 ALDH1A1 (0.54) MAPTKMT2AALDH1A1MEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6657083-B2 Photographic couplers; acylation amine group in position 2 EASTMAN KODAK COMPANY 2003-12-02 US disclosed
US-6613943-B2 Intermediates for 4-substituted-2,5-diaminophenol derivatives as phenolic cyan couplers for color photography; deblocking the 2-acyl group by hydrolysis EASTMAN KODAK COMPANY 2003-09-02 US disclosed
US-20030109716-A1 5-ACYLAMINO-2-AMINO-4-SUBSTITUTED-PHENOL COMPOUNDS AND METHOD OF USING THEM EASTMAN KODAK COMPANY 2003-06-12 US disclosed
US-20030109753-A1 4-acylamino-2-hydroxy-5-substituted-acylanilide compounds and method of using them EASTMAN KODAK COMPANY 2003-06-12 US disclosed
EP-1316550-A1 6-Acylamino-5-substituted-benzoxazol-2-one compounds and method for using them EASTMAN KODAK COMPANY (US) 2003-06-04 EP disclosed
EP-1316544-A1 5-acylamino-2-amino-4-substituted-phenol compounds and method of using them EASTMAN KODAK COMPANY (US) 2003-06-04 EP disclosed
US-6525219-B1 Chemical intermediates for cyan dye forming couplers; deblocking, hydrolysis, acylation EASTMAN KODAK COMPANY 2003-02-25 US disclosed
US-6515176-B1 Disclosed is a 6-acylamino-5-substituted-benzoxazol-2-one compound having the structural formula I: Also disclosed is a method for forming a cyan dye-forming coupler from the above compound. The method and intermediate with a simplified EASTMAN KODAK COMPANY 2003-02-04 US disclosed
US-6482953-B1 2-benzyloxy-4-nitro-5-substituted-acylanilide compounds and method of using them EASTMAN KODAK COMPANY 2002-11-19 US disclosed
US-6482985-B1 2-benzyloxy-5-halo-acylanilide compounds and method of using them EASTMAN KODAK COMPANY 2002-11-19 US disclosed
US-6476202-B1 5-acylamino-2-arylazo, nitro, or nitroso-4-substituted-phenol compounds and method of using them EASTMAN KODAK COMPANY 2002-11-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030109753-A1 4-acylamino-2-hydroxy-5-substituted-acylanilide compounds and method of using them CBR3, AADAC, HAAO MGLL 2331/4885MAPT 4684/4885KMT2A 665/4885
US-20030109716-A1 5-ACYLAMINO-2-AMINO-4-SUBSTITUTED-PHENOL COMPOUNDS AND METHOD OF USING THEM AADAT, AAAS, ANXA7 MGLL 3314/4885MAPT 2670/4885KMT2A 447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.