SCHEMBL7169997

SCHEMBL7169997

COC(=O)N1C[C@@H]2CCC(CN(CC#N)Cc3ccccc3OC)CC2CC1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
GRIN2B Q13224 2/20 0.36
BCHE P06276 9/20 0.36
ACHE P22303 9/20 0.36
BRD4 O60885 1/20 0.35
TACR1 P25103 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7161639 0.89 PGR (0.35) CYP2D6
SCHEMBL7170649 0.89 LTC4S (0.37)
SCHEMBL7163823 0.88 PGR (0.40) SLC6A2SLC6A4CYP2D6
SCHEMBL7166478 0.84 AGTR2 (0.37)
SCHEMBL7170300 0.84 TAS2R14 (0.35) SMN1; SMN2ALDH1A1TAS2R14
SCHEMBL7141654 0.83 LTC4S (0.37) BRD4CYP2D6ALDH1A1TAS2R14
SCHEMBL7168153 0.80 GRIN2B (0.46) SMN1; SMN2GRIN2BBCHEACHEBRD4
SCHEMBL7170826 0.72 CXCR4 (0.40) GRIN2BCYP2D6
SCHEMBL7171997 0.71 CXCR4 (0.40) ALDH1A1
SCHEMBL6327750 0.71 TSHR (0.35) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082856-A1 ISOQUINOLINE-3-CARBOXYLIC ACID DERIVATIVES AS EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2003-10-09 WO disclosed