SCHEMBL7166478

SCHEMBL7166478

COC(=O)N1C[C@@H]2CCC(CN(CC#N)CCc3ccccc3)CC2CC1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 8/20 0.37
OPRM1 P35372 4/20 0.37
OPRK1 P41145 4/20 0.37
OPRD1 P41143 3/20 0.37
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
ACE P12821 5/20 0.35
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7161639 0.91 PGR (0.35) AGTR2ACE
SCHEMBL7141654 0.85 LTC4S (0.37) MEN1LMNAKMT2A
SCHEMBL7170300 0.84 TAS2R14 (0.35)
SCHEMBL7169997 0.84 SMN1; SMN2 (0.37)
SCHEMBL7170649 0.83 LTC4S (0.37) ACE
SCHEMBL7163823 0.82 PGR (0.40)
SCHEMBL7165958 0.79 AGTR2 (0.41) AGTR2ACEMEN1USP2LMNA
SCHEMBL7171997 0.77 CXCR4 (0.40) ACEMEN1USP2LMNAKMT2A
SCHEMBL6327750 0.72 TSHR (0.35)
SCHEMBL6484834 0.72 TACR1 (0.41) AGTR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082856-A1 ISOQUINOLINE-3-CARBOXYLIC ACID DERIVATIVES AS EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2003-10-09 WO disclosed