SCHEMBL717410

SCHEMBL717410

C1CCC2OCCNC2C1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.35
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
DRD3 P35462 1/20 0.33
PDK1 Q15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL937953 1.00 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
SCHEMBL8232360 1.00 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
SCHEMBL5946959 1.00 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
SCHEMBL937955 1.00 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
Bromide SCHEMBL28439253 0.98 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
Hydrochloric Acid SCHEMBL697063 0.98 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
Hydrochloric Acid SCHEMBL17314206 0.98 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
Hydrochloric Acid SCHEMBL17314204 0.98 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
Hydrochloric Acid SCHEMBL696758 0.98 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1
Hydrochloric Acid SCHEMBL697062 0.98 HRH4 (0.35) HRH4GRIN1GRIN2ADRD3PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 206 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025124571-A1 NMDA RECEPTOR ANTAGONIST AND USE THEREOF 斯莱普泰(上海)生物医药科技有限公司 2025-06-19 WO claimed
CN-1099747-A Benzylhydrazone derivatives, a process for production thereof, and agricultural and horticultural fungicides NIHON NOHYAKU CO LTD (JP) 1995-03-08 CN claimed
EP-0622355-A2 Benzylhydrazone derivates, a process for production thereof, and agricultural and horticultural fungicides NIHON NOHYAKU CO., LTD. (JP) 1994-11-02 EP claimed
CN-1088384-A Contain the agricultural fungicide and the application thereof of N-(benzyloxy of replacement) imine derivative NIHON NOHYAKU CO LTD (JP) 1994-06-29 CN claimed
CN-1049654-A N- (substituted benzyloxy) imine derivatives, process for their preparation, their use and methods of use NIHON NOHYAKU CO LTD (JP) 1991-03-06 CN claimed
EP-0414153-A1 N-(substituted benzyloxy)imine derivatives, process for the production thereof, use thereof, and method of use thereof NIHON NOHYAKU CO., LTD. (JP) 1991-02-27 EP claimed
US-20250223262-A1 SYNTHESIS OF MORPHINANS WITH REDUCED HERG ACTIVITY AND MOP BINDING TAROS CHEMICALS GMBH & CO. KG (DE) 2025-07-10 US disclosed
WO-2025124571-A1 NMDA RECEPTOR ANTAGONIST AND USE THEREOF 斯莱普泰(上海)生物医药科技有限公司 2025-06-19 WO disclosed
EP-4499223-A1 SYNTHESIS OF MORPHINANS WITH REDUCED HERG ACTIVITY AND MOP BINDING Heinrich-Heine-Universität Düsseldorf (DE) 2025-02-05 EP disclosed
WO-2023187099-A1 SYNTHESIS OF MORPHINANS WITH REDUCED HERG ACTIVITY AND MOP BINDING HEINRICH-HEINE-UNIVERSITÄT DÜSSELDORF (DE) 2023-10-05 WO disclosed
US-20230303573-A1 3-((Hetero-)Aryl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives Grünenthal GmbH (DE) 2023-09-28 US disclosed
EP-3571205-B1 THIENOPYRIMIDINE DERIVATIVE AND USE THEREOF IN MEDICINE SUNSHINE LAKE PHARMA CO LTD (CN) 2023-08-30 EP disclosed
US-20230183184-A1 3-(Carboxyethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives GRUENENTHAL GMBH (DE) 2023-06-15 US disclosed
US-4587336-A PARKINSON'S DISEASE ELI LILLY AND COMPANY (US) 1986-05-06 US disclosed
US-4552956-A DOPAMINE AGONISTS ELI LILLY AND COMPANY (US) 1985-11-12 US disclosed
EP-0061900-B1 MORPHOLINES JOHN WYETH & BROTHER LIMITED (GB) 1985-03-20 EP disclosed
EP-0061899-B1 MORPHOLINES JOHN WYETH & BROTHER LIMITED (GB) 1985-03-20 EP disclosed
US-4409218-A Analgesic method JOHN WYETH AND BROTHER LIMITED (GB) 1983-10-11 US disclosed
US-4387097-A Morpholines JOHN WYETH AND BROTHER LIMITED (GB) 1983-06-07 US disclosed
EP-0061899-A1 Morpholines JOHN WYETH & BROTHER LIMITED (GB) 1982-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303573-A1 3-((Hetero-)Aryl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives OPRK1, OPRD1, OPRL1 HRH4 1326/4885GRIN1 133/4885GRIN2A 22/4885
US-20230183184-A1 3-(Carboxyethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives OPRK1, OPRD1, PKD2 HRH4 2163/4885GRIN1 324/4885GRIN2A 80/4885
US-20250223262-A1 SYNTHESIS OF MORPHINANS WITH REDUCED HERG ACTIVITY AND MOP BINDING OPRM1, TRPM5, TRPM7 HRH4 1811/4885GRIN1 434/4885GRIN2A 267/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.