SCHEMBL7177971

SCHEMBL7177971

CC(C)CC1Nc2c(S(=O)(=O)Oc3ccccc3)ccc(N3CCN(C)CC3)c2NC1=O

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 15/20 0.35
LMNA P02545 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
EGFR P00533 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
OXTR P30559 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7673285 0.99 CCR5 (0.36) CCR5LMNACYP3A4CYP2D6CYP2C9
SCHEMBL7674864 0.64 LMNA (0.43) LMNACYP3A4CYP2D6MAPTMAPK1
SCHEMBL7170492 0.62 ALDH1A1 (0.46) LMNAMAPTKMT2A
Hydrochloric Acid SCHEMBL7669155 0.62 LMNA (0.37) LMNAMAPTMAPK1KMT2A
SCHEMBL17676992 0.58 KDM4E (0.59) LMNAMAPTMAPK1KMT2ATP53
SCHEMBL10326483 0.58 KDM4E (0.59) LMNAMAPTMAPK1KMT2ATP53
SCHEMBL10327021 0.58 KDM4E (0.59) LMNAMAPTMAPK1KMT2ATP53
SCHEMBL3124456 0.55 GAA (0.51)
SCHEMBL17867151 0.55 GAA (0.51)
SCHEMBL2864427 0.55 GAA (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657166-B1 Combination containing a quinoxaline and a nucleoside AVENTIS PHARMA GMBH (DE) 2003-04-09 EP disclosed
US-6369057-B1 VIRICIDES, IN PARTICULAR AGAINST RETROVIRUSES, HUMAN IMMUNODEFICIENCY VIRUS (HIV) AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-04-09 US disclosed
EP-0509398-B1 Quinoxalines, process for their preparation and their use AVENTIS PHARMA GMBH (DE) 2001-09-19 EP disclosed
EP-0657166-A1 Combination containing a quinoxaline and a nucleoside HOECHST AKTIENGESELLSCHAFT (DE) 1995-06-14 EP disclosed
EP-0509398-A1 Quinoxalines, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1992-10-21 EP disclosed