SCHEMBL718209

SCHEMBL718209

Cc1[nH]c(N)nc(=O)c1C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.39
PNP P00491 2/20 0.37
CYP3A4 P08684 1/20 0.37
BLM P54132 1/20 0.37
HSD17B10 Q99714 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
CYP1A2 P05177 1/20 0.35
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TYMP P19971 1/20 0.33
FABP6 P51161 1/20 0.33
BACE1 P56817 1/20 0.33
MAPT P10636 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14217450 0.81 TYMP (0.43) XDHPNPCYP3A4BLMHSD17B10
SCHEMBL172129 0.75 ALDH1A1 (0.37) ALDH1A1L3MBTL1MAPT
SCHEMBL8531415 0.74 KDM5B (0.33) XDHPNPCYP3A4BLMHSD17B10
SCHEMBL4070047 0.71 TYMS (0.38) XDHCYP3A4BLMNPSR1ALDH1A1
SCHEMBL9879126 0.70 L3MBTL1 (0.46) XDHPNPNPSR1L3MBTL1BACE1
SCHEMBL9965294 0.70 HSD17B10 (0.46) PNPCYP3A4HSD17B10NPSR1CYP1A2
SCHEMBL27942625 0.70 MAPK1 (0.39) XDHHSD17B10NPSR1ALDH1A1BACE1
SCHEMBL11988254 0.69 HSD17B10 (0.45) CYP3A4HSD17B10NPSR1CYP1A2ALDH1A1
SCHEMBL28460640 0.69 HSD17B10 (0.42) CYP3A4HSD17B10NPSR1CYP1A2ALDH1A1
SCHEMBL215067 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114716961-B Self-complementary quadruple hydrogen bond supermolecule hot melt adhesive and synthesis method thereof 郑州大学 2023-06-23 CN disclosed
CN-114716961-A Self-complementary quadruple hydrogen bond supramolecular hot melt adhesive and synthesis method thereof 郑州大学 2022-07-08 CN disclosed
US-20120302587-A1 RHO-KINASE INHIBITORS NAGARAHNAM DHANAPALAN (US) 2012-11-29 US disclosed
EP-1470121-B1 PYRIMIDINE DERIVATIVES AS RHO-KINASE INHIBITORS BAYER HEALTHCARE LLC (US) 2012-07-11 EP disclosed
US-20120053179-A1 Rho-Kinase Inhibitors NAGARATHNAM DHANAPALAN (US) 2012-03-01 US disclosed
EP-1470122-B1 RHO-KINASE INHIBITORS BAYER PHARMACEUTICALS CORP (US) 2007-12-19 EP disclosed
US-20050209261-A1 Rho-kinase inhibitors BAYER HEALTHCARE LLC 2005-09-22 US disclosed
US-6943172-B2 Rho-kinase inhibitors BAYER PHARMACEUTICALS CORPORATION (US) 2005-09-13 US disclosed
US-20050192304-A1 Rho-kinase inhibitors BAYER HEALTHCARE LLC 2005-09-01 US disclosed
US-6924290-B2 Rho-kinase inhibitors BAYER PHARMACEUTICALS CORPORATION (US) 2005-08-02 US disclosed
EP-1470122-A1 RHO-KINASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-10-27 EP disclosed
EP-1470121-A1 PYRIMIDINE DERIVATIVES AS RHO-KINASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-10-27 EP disclosed
US-20040002508-A1 Antitumor agents; anticancer agents; sexual disorders; cardiovascular disorders BAYER CORPORATION 2004-01-01 US disclosed
US-20040002507-A1 Rho-kinase inhibitors BAYER CORPORATION (US) 2004-01-01 US disclosed
WO-2003062227-A1 RHO-KINASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-31 WO disclosed
WO-2003062225-A1 PYRIMIDINE DERIVATIVES AS RHO-KINASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040002507-A1 Rho-kinase inhibitors CIT, ROCK1, ROCK2 XDH 598/4885PNP 1050/4885CYP3A4 2878/4885
US-20120053179-A1 Rho-Kinase Inhibitors CIT, ROCK1, ROCK2 XDH 598/4885PNP 1050/4885CYP3A4 2878/4885
US-20050209261-A1 Rho-kinase inhibitors CIT, ROCK1, ROCK2 XDH 598/4885PNP 1050/4885CYP3A4 2878/4885
US-20040002508-A1 Antitumor agents; anticancer agents; sexual disorders; cardiovascular disorders CIT, ROCK1, RHOT2 XDH 564/4885PNP 1179/4885CYP3A4 2456/4885
US-20120302587-A1 RHO-KINASE INHIBITORS CIT, ROCK1, ROCK2 XDH 598/4885PNP 1050/4885CYP3A4 2878/4885
US-20050192304-A1 Rho-kinase inhibitors CIT, ROCK1, ROCK2 XDH 598/4885PNP 1050/4885CYP3A4 2878/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.