SCHEMBL7183929

SCHEMBL7183929

CC(=O)OC[C@@H](C)Nc1ncc(C#N)cc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
GLA P06280 2/20 0.39
HCAR3 P49019 1/20 0.36
JAK2 O60674 2/20 0.35
JAK3 P52333 2/20 0.35
VCAM1 P19320 1/20 0.35
MTOR P42345 1/20 0.34
PLK1 P53350 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
PKM P14618 1/20 0.34
IRAK4 Q9NWZ3 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185895 0.84 ALDH1A1 (0.44) ALDH1A1GLAJAK2JAK3VCAM1
SCHEMBL7182989 0.82 MAPK8 (0.38) IRAK4
SCHEMBL7191686 0.80 L3MBTL1 (0.45) ALDH1A1LMNAMAPTPKM
SCHEMBL7190961 0.80 HCAR3 (0.53) ALDH1A1HCAR3VCAM1LMNAMAPT
SCHEMBL7184178 0.80 HCAR3 (0.53) ALDH1A1HCAR3VCAM1LMNAMAPT
SCHEMBL30989701 0.73 VCAM1 (0.47) ALDH1A1JAK2JAK3VCAM1LMNA
SCHEMBL25887391 0.73 VCAM1 (0.47) ALDH1A1JAK2JAK3VCAM1LMNA
SCHEMBL26914382 0.73 GLA (0.41) ALDH1A1GLAJAK2JAK3VCAM1
SCHEMBL26914255 0.73 GLA (0.41) ALDH1A1GLAJAK2JAK3VCAM1
SCHEMBL26914256 0.73 GLA (0.41) ALDH1A1GLAJAK2JAK3VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6582351-B1 Benzimidazole heterocyclic compounds having pharmacological activities, and their use as a medicament for treatment or prevention of diseases mediated by cGMP-PDE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-06-24 US disclosed