SCHEMBL7188673

SCHEMBL7188673

CC[C@@H](COC(C)=O)Nc1ccc(C#N)cc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HCAR3 P49019 1/20 0.34
MAP2K1 Q02750 4/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
MTOR P42345 1/20 0.33
GSK3B P49841 1/20 0.33
PRKDC P78527 1/20 0.33
KCNH2 Q12809 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7190795 1.00 GAA (0.39) GAAKDM4EALDH1A1HCAR3MAP2K1
SCHEMBL7183015 0.85 KDM4E (0.44) GAAKDM4EALDH1A1HCAR3MAP2K1
SCHEMBL7185647 0.85 KDM4E (0.44) GAAKDM4EALDH1A1HCAR3MAP2K1
SCHEMBL7189685 0.83 HCAR3 (0.53) KDM4EALDH1A1HCAR3LMNATDP1
SCHEMBL7185695 0.83 HCAR3 (0.53) KDM4EALDH1A1HCAR3LMNATDP1
SCHEMBL7183531 0.73 ALDH1A1 (0.41) GAAKDM4EALDH1A1MAP2K1ABCC9
SCHEMBL7191231 0.73 PTGER4 (0.48) GAAKDM4EALDH1A1
SCHEMBL7387168 0.70 KDM4E (0.51) GAAKDM4EALDH1A1POLB
SCHEMBL15595142 0.70 LMNA (0.44) GAAKDM4EALDH1A1MAP2K1GPR35
SCHEMBL2339309 0.70 KDM4E (0.54) GAAKDM4EALDH1A1ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6582351-B1 Benzimidazole heterocyclic compounds having pharmacological activities, and their use as a medicament for treatment or prevention of diseases mediated by cGMP-PDE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-06-24 US disclosed