SCHEMBL7198022

SCHEMBL7198022

CCOC(=O)N(C(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](C)N)C(C)C)[C@@H](CC(=O)OC(C)(C)C)CC(OCC)OCC

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.38
CTSD P07339 3/20 0.37
REN P00797 3/20 0.37
CASP1 P29466 3/20 0.36
HLA-DRB1 P01911 1/20 0.35
CASP3 P42574 2/20 0.35
CASP7 P55210 1/20 0.35
BACE1 P56817 2/20 0.35
BACE2 Q9Y5Z0 2/20 0.35
MMP1 P03956 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
CASP9 P55211 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5686897 0.86 CTSD (0.37) OPRD1CTSD
SCHEMBL5689430 0.85 OPRD1 (0.40) OPRD1CTSDCASP1
SCHEMBL5686592 0.80 OPRD1 (0.46) OPRD1RENCASP1HLA-DRB1CASP3
SCHEMBL5686579 0.80 CTSD (0.38) OPRD1CTSD
SCHEMBL7198017 0.79 REN (0.46) OPRD1CTSDRENCASP1HLA-DRB1
SCHEMBL5689425 0.76 CASP1 (0.49) OPRD1CTSDRENCASP1HLA-DRB1
SCHEMBL5686711 0.73 CTSD (0.36) OPRD1CTSDBACE1
SCHEMBL5686675 0.73 CASP1 (0.47) OPRD1RENCASP1CASP3CASP7
SCHEMBL5686901 0.72 REN (0.46) CTSDRENCASP1HLA-DRB1CTSS
SCHEMBL5686703 0.72 REN (0.42) CTSDRENBACE1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6593300-B1 Inhibitors of the interleukin-1 beta converting enzyme GYOGYSZERKUTATO INTEZET KFT. (HU) 2003-07-15 US disclosed
EP-0979241-A1 (3R)-3-AMINO-4-CARBOXYBUTYRALDEHYDE DERIVATIVES INHIBITING THE RELEASE OF INTERLEUKIN-1/BETA GYOGYSZERKUTATO INTEZET KFT. (HU) 2000-02-16 EP disclosed
WO-1998049189-A1 (3R)-3-AMINO-4-CARBOXYBUTYRALDEHYDE DERIVATIVES INHIBITING THE RELEASE OF INTERLEUKIN-1/BETA Gyógyszerkutató Intézet Kft. (HU) 1998-11-05 WO disclosed