SCHEMBL7201516

SCHEMBL7201516

CC(=O)N(N)c1cccc(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.48
PARP1 P09874 1/20 0.46
HSD17B1 P14061 5/20 0.44
HSD17B2 P37059 5/20 0.44
HSD17B10 Q99714 2/20 0.43
SIGMAR1 Q99720 1/20 0.42
ALDH1A1 P00352 5/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
PAX8 Q06710 2/20 0.42
JAK2 O60674 1/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 2/20 0.42
APAF1 O14727 1/20 0.42
TDP2 O95551 1/20 0.42
NFKB1 P19838 1/20 0.42
CASP3 P42574 1/20 0.42
BLM P54132 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27430312 0.80 MEN1 (0.44) LMNAPARP1HSD17B1HSD17B2HSD17B10
SCHEMBL9998812 0.80 CRHBP (0.53) LMNAPARP1HSD17B1HSD17B2HSD17B10
SCHEMBL10441683 0.79 HTR3E (0.50) LMNAPARP1ALDH1A1NPC1RAB9A
SCHEMBL28980326 0.79 MTNR1A (0.47) LMNAPARP1ALDH1A1NPC1RAB9A
SCHEMBL29279420 0.79 TP53 (0.43) LMNAPARP1HSD17B1HSD17B2SIGMAR1
SCHEMBL30545032 0.79 HSD17B1 (0.41) LMNAPARP1HSD17B1HSD17B2SIGMAR1
SCHEMBL28490022 0.79 CYP3A4 (0.55) PARP1HSD17B1HSD17B2ALDH1A1NPC1
SCHEMBL29674755 0.78 HSD17B1 (0.57) LMNAHSD17B1HSD17B2HSD17B10SIGMAR1
SCHEMBL10836221 0.78 MEN1 (0.53) LMNAPARP1HSD17B1HSD17B2HSD17B10
SCHEMBL2531803 0.78 HSD17B1 (0.57) LMNAHSD17B1HSD17B2HSD17B10SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894326-B 2, 3-Hydrogen substituted aminoindole derivative, preparation method and application thereof 佛山大学 2025-02-11 CN disclosed
CN-115894326-A 2,3-hydrogen substituted aminoindole derivative, preparation method and application thereof 佛山科学技术学院 2023-04-04 CN disclosed
CN-109467528-B Synthesis method of 1-aminoindole derivative 佛山科学技术学院 2020-11-06 CN disclosed
CN-104262284-A 2-amino-1, 3, 4-oxadiazole compound and preparation method thereof UNIV SHANGHAI 2015-01-07 CN disclosed
US-6656910-B2 Serine protease inhibitors CORTECH, INC. 2003-12-02 US disclosed
US-6656911-B2 Oxadiazole ring structure peptoids which are useful as inhibitors of serine proteases CORTECH, INC. 2003-12-02 US disclosed
US-20030203851-A1 Substituted oxadiazole, peptoids which are useful for treating adult respiratory distress syndrome, septic shock and myocardial ischemia-reperfusion injury CORTECH, INC. 2003-10-30 US disclosed
US-6608175-B2 Oxadiazole, thiadiazoles or triazole metal derivatives reacted with an amine containing aldehyde, deprotecting, coupling with an acid and oxidizing to create substituted oxadiazole, thiadiazole or triazole peptoids CORTECH, INC. 2003-08-19 US disclosed
US-20030060418-A1 Serine protease inhibitors CORTECH, INC. 2003-03-27 US disclosed
US-20020119985-A1 Serine protease inhibitors CORTECH, INC. 2002-08-29 US disclosed
US-6001811-A TREATMENT OF ADULT RESPIRATORY DISTRESS SYNDROME, SEPSIS, MULTIPLE ORGAN FAILURE CORTECH INC. (US) 1999-12-14 US disclosed
US-5998379-A USEFUL AS INHIBITORS OF SERINE PROTEASES, IN PARTICULAR HUMAN NEUTROPHIL ELASTASE, TREATMENT OF ADULT RESPIRATORY DISTRESS SYNDROME, SEPTIC SHOCK, AND MYOCARDIAL ISCHEMIA-REPERFUSION INJURY CORTECH INC. (US) 1999-12-07 US disclosed
WO-1999054317-A1 CYSTEINE PROTEASE INHIBITORS CORTECH INC. (US) 1999-10-28 WO disclosed
WO-1998049190-A9 SUBSTITUTED OXADIAZOLE CYSTEINE PROTEASE INHIBITORS CORTECH INC (US) 1999-04-15 WO disclosed
US-5891852-A Serine protease inhibitors-cycloheptane derivatives CORTECH, INC. (US) 1999-04-06 US disclosed
US-5869455-A SUBSTITUTED OXADIAZOLE, THIADIAZOLE AND TRIAZOLE PEPTOIDS WHICH ARE USEFUL AS INHIBITORS OF HUMAN NEUTROPHIL ELASTASE CORTECH, INC. (US) 1999-02-09 US disclosed
US-5861380-A OXADIAZOLE, THIADIAZOLE AND TRIAZOLE PEPTOIDS AS INHIBITORS OF HUMAN NEUTROPHIL ELASTASE; ADULT RESPIRATORY DISTRESS SYNDROME; ANTIARTHRITIC,-INFLAMMATORY,-ISCHEMIC,-TUMOR AND -CARCINOGENIC AGENTS AND OTHER HNE-MEDIATED CONDITIONS CORTECH, INC. (US) 1999-01-19 US disclosed
WO-1998049190-A2 SUBSTITUTED OXADIAZOLE CYSTEINE PROTEASE INHIBITORS CORTECH, INC. (US) 1998-11-05 WO disclosed
US-5807829-A RESPIRATORY SYSTEM DISORDERS; SESPIC SHOCK; ORGAN FAILURE CORTECH, INC. (US) 1998-09-15 US disclosed
US-5801148-A Serine protease inhibitors-proline analogs CORTECH, INC. (US) 1998-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020119985-A1 Serine protease inhibitors PRSS1, SERPINB1, SERPINE1 LMNA 4083/4885PARP1 1633/4885HSD17B1 1018/4885
US-20030203851-A1 Substituted oxadiazole, peptoids which are useful for treating adult respiratory distress syndrome, septic shock and myocardial ischemia-reperfusion injury TNNI3, PEPD, STK35 LMNA 4508/4885PARP1 2821/4885HSD17B1 746/4885
US-20030060418-A1 Serine protease inhibitors PRSS1, SERPINB1, SERPINE1 LMNA 4083/4885PARP1 1633/4885HSD17B1 1018/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.