SCHEMBL7208577

SCHEMBL7208577

NC(=O)C1OC(c2cccnc2)CC1(NS(=O)(=O)c1ccc(OCc2ccc(Cl)cc2F)cc1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 9/20 0.39
MMP1 P03956 4/20 0.39
ADAMTS5 Q9UNA0 3/20 0.38
MMP13 P45452 1/20 0.37
ADAMTS7 Q9UKP4 1/20 0.35
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7213016 0.82 ADAMTS5 (0.51) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7212988 0.81 MMP1 (0.41) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7207012 0.80 MMP13 (0.49) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7208565 0.79 MMP1 (0.49) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7214339 0.78 MMP1 (0.40) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7214304 0.77 MMP1 (0.37) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7212996 0.74 MMP1 (0.42) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7209169 0.74 MMP1 (0.43) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL7213084 0.72 ADAMTS5 (0.40) ADAM17MMP1ADAMTS5MMP13ADAMTS7
SCHEMBL5492928 0.71 ADAMTS5 (0.64) ADAM17MMP1ADAMTS5MMP13ADAMTS7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed